SCHEMBL10667334

SCHEMBL10667334

CNCCc1csc2ccc(Br)cc12

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.59
CA2 P00918 1/20 0.52
CHRNB2 P17787 1/20 0.49
CHRNA7 P36544 1/20 0.49
CHRNA4 P43681 1/20 0.49
MTNR1A P48039 10/20 0.47
MTNR1B P49286 4/20 0.47
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
TAAR1 Q96RJ0 3/20 0.43
CHEK1 O14757 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10668808 0.83 CA2 (0.54) CYP2A6CA2MTNR1AMTNR1B
SCHEMBL6075756 0.82 MTNR1A (0.72) CYP2A6CA2MTNR1AMTNR1BHDAC10
SCHEMBL6076645 0.81 MTNR1A (0.72) CYP2A6CA2MTNR1AMTNR1BHDAC10
SCHEMBL25987518 0.81 KDM4E (0.52) CYP2A6MTNR1AMTNR1B
SCHEMBL31588788 0.80 CYP2A6 (0.67) CYP2A6CA2MTNR1AMTNR1BHDAC10
SCHEMBL25030227 0.79 MTNR1A (0.70) MTNR1AMTNR1B
SCHEMBL8547530 0.79 CYP2A6 (0.75) CYP2A6CA2MTNR1AMTNR1BHDAC10
SCHEMBL6075680 0.78 MTNR1A (0.66) CYP2A6CA2MTNR1AMTNR1BHDAC10
SCHEMBL8551337 0.78 CYP2A6 (0.59) CYP2A6CA2MTNR1AMTNR1BHDAC10
SCHEMBL15985408 0.78 MTNR1A (0.47) CYP2A6MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4737495-A ANTIALLERGENS, ANTISCHEMIC, HYPOTENSIVE AGENTS DR. KARL TOMAE, GMBH (DE) 1988-04-12 US disclosed
EP-0204349-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1986-12-10 EP disclosed