SCHEMBL10667474

SCHEMBL10667474

NC(Cc1cc(Cl)c(O)c(Br)c1)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 4/20 0.52
THRA P10827 2/20 0.52
PPARG P37231 2/20 0.52
GRIA2 P42262 1/20 0.49
SIRT5 Q9NXA8 1/20 0.48
HSD17B10 Q99714 5/20 0.47
USP2 O75604 4/20 0.47
ALOX15 P16050 4/20 0.47
SLC7A5 Q01650 3/20 0.47
ADORA3 P0DMS8 3/20 0.47
TDP1 Q9NUW8 3/20 0.47
PTGS1 P23219 2/20 0.47
PTGS2 P35354 2/20 0.47
KDM4E B2RXH2 2/20 0.47
RECQL P46063 2/20 0.47
HIF1A Q16665 2/20 0.47
EGFR P00533 1/20 0.47
LCK P06239 1/20 0.47
FYN P06241 1/20 0.47
HTR2A P28223 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10667480 1.00 THRB (0.52) THRBTHRAPPARGGRIA2SIRT5
SCHEMBL2122000 0.89 SLC7A5 (0.55) THRBTHRAPPARGGRIA2SIRT5
SCHEMBL31083609 0.89 SLC7A5 (0.55) THRBTHRAPPARGGRIA2SIRT5
SCHEMBL2121998 0.89 SLC7A5 (0.55) THRBTHRAPPARGGRIA2SIRT5
Dibromotyrosine SCHEMBL145218 0.89 THRB (0.58) THRBTHRAPPARGGRIA2SIRT5
Dibromotyrosine SCHEMBL838919 0.89 THRB (0.58) THRBTHRAPPARGGRIA2SIRT5
Dibromotyrosine SCHEMBL145219 0.89 THRB (0.58) THRBTHRAPPARGGRIA2SIRT5
Dibromotyrosine SCHEMBL29399010 0.87 THRB (0.57) THRBTHRAPPARGGRIA2SIRT5
Hydrochloric Acid SCHEMBL16007570 0.87 GRIA2 (0.53) THRBTHRAPPARGGRIA2SIRT5
Hydrochloric Acid SCHEMBL16007571 0.87 GRIA2 (0.53) THRBTHRAPPARGGRIA2SIRT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4745124-A THIO/ESTER PEPTIDES UNIVERSITY OF MIAMI (US) 1988-05-17 US disclosed
US-4690936-A AMINO ACIDS, THIOESTER LINKAGE; ANGIOTENSIN INHIBITORS UNIVERSITY OF MIAMI (US) 1987-09-01 US disclosed