SCHEMBL10668604

SCHEMBL10668604

COc1nc2nc(S(=O)(=O)Nc3c(F)cccc3C(=O)OC(C)C)nn2cc1C

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
NPC1 O15118 1/20 0.31
EDNRA P25101 2/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10660656 0.92 TSHR (0.34) TSHRNPC1EDNRA
SCHEMBL10664390 0.92 KMT2A (0.36) TSHRKMT2A
SCHEMBL10664359 0.90 CCR4 (0.34) TSHR
SCHEMBL10666211 0.89 THRB (0.33) TSHR
SCHEMBL10663320 0.89 TSHR (0.42) TSHRNPC1KMT2A
SCHEMBL10667939 0.86 CA12 (0.31) TSHR
SCHEMBL10662520 0.84 MAPT (0.34)
SCHEMBL10663456 0.84 TSHR (0.38) TSHRKMT2A
SCHEMBL10663171 0.84 NPC1 (0.30) NPC1
SCHEMBL9833287 0.84 LMNA (0.32) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4755212-A Novel substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonamides and compositions and method for inhibiting pollen formation in corn THE DOW CHEMICAL COMPANY (US) 1988-07-05 US disclosed
US-4741764-A SUPPRESSION OF NITRIFICATION OF AMMONIUM NITROGEN IN THE SOIL THE DOW CHEMICAL COMPANY (US) 1988-05-03 US disclosed
US-4740233-A Substituted 1,2,4-triazolo[1,5-a]-pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1988-04-26 US disclosed