SCHEMBL10677643

SCHEMBL10677643

O=c1cc(-c2ccccc2)oc2cc(OC3CCCNCC3)ccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.55
TNKS O95271 2/20 0.55
TP53 P04637 2/20 0.52
CYP3A4 P08684 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
MEN1 O00255 1/20 0.52
LMNA P02545 1/20 0.52
MAPT P10636 1/20 0.52
KMT2A Q03164 1/20 0.52
ROCK1 Q13464 2/20 0.51
MAOB P27338 2/20 0.48
CA12 O43570 2/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
ABCB1 P08183 2/20 0.48
CYP1B1 Q16678 2/20 0.48
CA9 Q16790 2/20 0.48
AKR1B10 O60218 1/20 0.48
CYP1A2 P05177 1/20 0.48
CALM1 P0DP23 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10681161 0.93 ABCB1 (0.56) TNKSTP53CYP3A4MAPTROCK1
SCHEMBL10683812 0.81 CYP19A1 (0.54) CYP19A1TNKSTP53CYP3A4SMN1; SMN2
SCHEMBL10680679 0.81 MAOA (0.58) CYP19A1TNKSTP53CYP3A4SMN1; SMN2
SCHEMBL10683600 0.80 AR (0.55) TP53CYP3A4SMN1; SMN2MEN1MAPT
SCHEMBL10683624 0.79 NPC1 (0.57) TP53CYP3A4SMN1; SMN2MEN1MAPT
SCHEMBL10684459 0.78 ABCG2 (0.53) CYP19A1TNKSSIGMAR1ABCG2
SCHEMBL10682295 0.76 CYP3A4 (0.64) CYP19A1TNKSTP53CYP3A4SMN1; SMN2
SCHEMBL10681965 0.76 MEN1 (0.57) CYP19A1TNKSTP53CYP3A4SMN1; SMN2
SCHEMBL10679051 0.75 CYP19A1 (0.51) CYP19A1TNKSTP53CYP3A4SMN1; SMN2
SCHEMBL10680511 0.74 ROCK1 (0.49) TP53CYP3A4SMN1; SMN2MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4780478-A Aminopropoxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 1988-10-25 US disclosed
US-4508732-A Basic ethers useful as antidepressant agents MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1985-04-02 US disclosed
EP-0031885-B1 BASIC ETHERS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION MERCK PATENT GmbH (DE) 1984-06-27 EP disclosed
US-4376123-A Hexahydroazepinyloxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1983-03-08 US disclosed
EP-0031885-A1 Basic ethers, pharmaceutical compositions containing them and process for their preparation MERCK PATENT GmbH (DE) 1981-07-15 EP disclosed