SCHEMBL10684459

SCHEMBL10684459

O=c1cc(-c2ccccc2)oc2cc(OCC3CCCNC3)ccc12

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 3/20 0.53
MAP2K1 Q02750 1/20 0.53
SIGMAR1 Q99720 6/20 0.53
TNKS O95271 1/20 0.52
CYP19A1 P11511 1/20 0.52
KDM4E B2RXH2 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10677317 0.93 KDM4E (0.54) ABCG2SIGMAR1KDM4E
SCHEMBL10684580 0.82 SIGMAR1 (0.52) ABCG2SIGMAR1KDM4E
SCHEMBL10682290 0.81 MAOA (0.67) SIGMAR1TNKSCYP19A1
SCHEMBL10682013 0.80 MAP2K1 (0.54) MAP2K1KDM4E
SCHEMBL10683812 0.79 CYP19A1 (0.54) ABCG2SIGMAR1TNKSCYP19A1KDM4E
SCHEMBL10486553 0.78 TNKS (0.61) ABCG2SIGMAR1TNKSCYP19A1KDM4E
SCHEMBL10682295 0.78 CYP3A4 (0.64) ABCG2SIGMAR1TNKSCYP19A1KDM4E
SCHEMBL10677643 0.78 CYP19A1 (0.55) ABCG2SIGMAR1TNKSCYP19A1
SCHEMBL10681965 0.77 MEN1 (0.57) TNKSCYP19A1
SCHEMBL10679051 0.77 CYP19A1 (0.51) ABCG2SIGMAR1TNKSCYP19A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4780478-A Aminopropoxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 1988-10-25 US disclosed
US-4508732-A Basic ethers useful as antidepressant agents MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1985-04-02 US disclosed
EP-0031885-B1 BASIC ETHERS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION MERCK PATENT GmbH (DE) 1984-06-27 EP disclosed
US-4376123-A Hexahydroazepinyloxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1983-03-08 US disclosed
EP-0031885-A1 Basic ethers, pharmaceutical compositions containing them and process for their preparation MERCK PATENT GmbH (DE) 1981-07-15 EP disclosed