SCHEMBL10679371

SCHEMBL10679371

CC(Oc1cccc2oc(-c3ccccc3)cc(=O)c12)C1CCCNC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.53
CYP3A4 P08684 5/20 0.53
ALDH1A1 P00352 4/20 0.53
TP53 P04637 4/20 0.53
MAPT P10636 4/20 0.53
KDM4E B2RXH2 3/20 0.53
HSD17B10 Q99714 2/20 0.53
HPGD P15428 1/20 0.53
ABCB1 P08183 4/20 0.45
SIGMAR1 Q99720 5/20 0.44
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
ABCG2 Q9UNQ0 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
LMNA P02545 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10682524 0.87 AR (0.49) ARCYP3A4ALDH1A1TP53MAPT
SCHEMBL10682295 0.82 CYP3A4 (0.64) CYP3A4ALDH1A1TP53MAPTKDM4E
SCHEMBL10681870 0.82 MAPT (0.54) CYP3A4ALDH1A1TP53MAPTKDM4E
SCHEMBL10682542 0.80 MAPT (0.41) CYP3A4ALDH1A1TP53MAPTKDM4E
SCHEMBL9138586 0.79 AR (0.72) ARCYP3A4ALDH1A1TP53MAPT
SCHEMBL10681056 0.79 CYP3A4 (0.54) ARCYP3A4ALDH1A1TP53MAPT
SCHEMBL10684580 0.78 SIGMAR1 (0.52) ARCYP3A4ALDH1A1TP53MAPT
SCHEMBL10686049 0.77 CYP3A4 (0.51) ARCYP3A4ALDH1A1TP53MAPT
SCHEMBL10683600 0.76 AR (0.55) ARCYP3A4ALDH1A1TP53MAPT
SCHEMBL11651074 0.75 CYP3A4 (0.69) ARCYP3A4ALDH1A1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4780478-A Aminopropoxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 1988-10-25 US disclosed
US-4508732-A Basic ethers useful as antidepressant agents MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1985-04-02 US disclosed
US-4376123-A Hexahydroazepinyloxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1983-03-08 US disclosed