SCHEMBL10684580

SCHEMBL10684580

O=c1cc(-c2ccccc2)oc2cccc(OCC3CCCNC3)c12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.52
AR P10275 4/20 0.52
ALDH1A1 P00352 4/20 0.52
CYP3A4 P08684 3/20 0.52
KDM4E B2RXH2 3/20 0.52
MAPT P10636 2/20 0.52
TP53 P04637 2/20 0.52
HSD17B10 Q99714 2/20 0.52
HPGD P15428 2/20 0.52
BCHE P06276 1/20 0.50
ACHE P22303 1/20 0.50
IKBKB O14920 1/20 0.47
CHUK O15111 1/20 0.47
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
CYP1A1 P04798 1/20 0.44
CYP1A2 P05177 1/20 0.44
PKM P14618 1/20 0.44
ALOX15 P16050 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10684459 0.82 ABCG2 (0.53) SIGMAR1KDM4EABCG2
SCHEMBL10677317 0.81 KDM4E (0.54) SIGMAR1ALDH1A1KDM4EMAPTNPC1
SCHEMBL10679358 0.81 SIGMAR1 (0.59) SIGMAR1ARALDH1A1CYP3A4KDM4E
SCHEMBL10679105 0.79 IKBKB (0.48) IKBKBCHUKCHRNB2CHRNA4CHRNB4
SCHEMBL10681056 0.79 CYP3A4 (0.54) SIGMAR1ARALDH1A1CYP3A4KDM4E
SCHEMBL9205310 0.78 AR (0.61) SIGMAR1ARALDH1A1CYP3A4KDM4E
SCHEMBL10679371 0.78 AR (0.53) SIGMAR1ARALDH1A1CYP3A4KDM4E
SCHEMBL10683600 0.78 AR (0.55) SIGMAR1ARALDH1A1CYP3A4KDM4E
SCHEMBL10682524 0.77 AR (0.49) SIGMAR1ARALDH1A1CYP3A4KDM4E
SCHEMBL10686049 0.77 CYP3A4 (0.51) SIGMAR1ARALDH1A1CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4780478-A Aminopropoxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 1988-10-25 US disclosed
US-4508732-A Basic ethers useful as antidepressant agents MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1985-04-02 US disclosed
EP-0031885-B1 BASIC ETHERS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION MERCK PATENT GmbH (DE) 1984-06-27 EP disclosed
US-4376123-A Hexahydroazepinyloxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1983-03-08 US disclosed
EP-0031885-A1 Basic ethers, pharmaceutical compositions containing them and process for their preparation MERCK PATENT GmbH (DE) 1981-07-15 EP disclosed