SCHEMBL10679398

SCHEMBL10679398

CCCC(N)=CC(=O)OC(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.40
HCAR2 Q8TDS4 1/20 0.39
TSHR P16473 1/20 0.33
ALDH1A1 P00352 2/20 0.32
CYP3A4 P08684 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CA12 O43570 1/20 0.32
AKR1B10 O60218 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
AKR1B1 P15121 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
CTSD P07339 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10679395 1.00 LMNA (0.40) LMNAHCAR2TSHRALDH1A1CYP3A4
SCHEMBL10684921 0.89 LMNA (0.46) LMNAHCAR2ALDH1A1CYP3A4TDP1
SCHEMBL10684914 0.89 LMNA (0.46) LMNAHCAR2ALDH1A1CYP3A4TDP1
SCHEMBL10683996 0.84 HCAR2 (0.42) LMNAHCAR2TSHRALDH1A1CYP3A4
SCHEMBL10683990 0.84 HCAR2 (0.42) LMNAHCAR2TSHRALDH1A1CYP3A4
SCHEMBL10679402 0.84 LMNA (0.30) LMNA
SCHEMBL10679390 0.84 LMNA (0.30) LMNA
SCHEMBL15482671 0.78 LMNA (0.41) LMNAHCAR2TSHRALDH1A1CYP3A4
SCHEMBL13468460 0.78 LMNA (0.41) LMNAHCAR2TSHRALDH1A1CYP3A4
SCHEMBL5452972 0.78 HCAR2 (0.39) HCAR2TSHRALDH1A1CYP3A4CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4761420-A CARDIOVASCULAR DISORDERS LABORATOIRES SYNTEX S.A. (FR) 1988-08-02 US disclosed
EP-0249245-A2 Antihypertensive dihydropyridine derivatives LABORATOIRES SYNTEX S.A. (FR) 1987-12-16 EP disclosed