SCHEMBL10679484

SCHEMBL10679484

CCN(CC)C(=O)CCc1c[nH]c2ccc(OC)cc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.64
CYP2D6 P10635 3/20 0.62
KMT2A Q03164 3/20 0.62
MTNR1A P48039 9/20 0.61
MTNR1B P49286 7/20 0.60
CYP1A2 P05177 3/20 0.60
KDM4E B2RXH2 2/20 0.60
HTR2B P41595 2/20 0.60
BLM P54132 2/20 0.60
PMP22 Q01453 2/20 0.60
MEN1 O00255 1/20 0.60
ALDH1A1 P00352 1/20 0.60
CYP1A1 P04798 1/20 0.60
MPO P05164 1/20 0.60
CYP3A4 P08684 1/20 0.60
HPGD P15428 1/20 0.60
NQO2 P16083 1/20 0.60
RAB9A P51151 1/20 0.60
CYP1B1 Q16678 1/20 0.60
NOTUM Q6P988 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24723377 0.88 KDM4E (0.70) HTR1ACYP2D6KMT2AMTNR1AMTNR1B
SCHEMBL4619391 0.84 CYP2D6 (0.64) HTR1ACYP2D6KMT2AMTNR1AMTNR1B
SCHEMBL3024961 0.83 KDM4E (0.75) HTR1ACYP2D6KMT2AMTNR1AMTNR1B
SCHEMBL4889276 0.83 MTNR1A (0.70) HTR1ACYP2D6KMT2AMTNR1AMTNR1B
SCHEMBL10671995 0.82 MTNR1A (0.58) HTR1AKMT2AMTNR1AMTNR1BHTR2B
SCHEMBL3018752 0.82 MTNR1A (0.70) HTR1ACYP2D6KMT2AMTNR1AMTNR1B
SCHEMBL5085972 0.80 KMT2A (0.65) HTR1ACYP2D6KMT2AMTNR1AMTNR1B
SCHEMBL8292283 0.80 CYP2D6 (0.68) HTR1ACYP2D6KMT2AMTNR1AMTNR1B
SCHEMBL10674520 0.79 ALDH1A1 (0.85) HTR1ACYP2D6KMT2ACYP1A2MEN1
SCHEMBL10670286 0.79 MTNR1A (0.71) HTR1ACYP2D6KMT2AMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4788204-A TRANQUILIZERS; ANTICONVULSANTS; ANGINA AND IMMUNODIFICIENCY TREATMENTS RHONE-POULENC SANTE (FR) 1988-11-29 US disclosed
US-4788199-A ANXIOLYTICS, ANTICONVULSANTS, ANTIANGINA AGENTS RHONE-POULENC SANTE (FR) 1988-11-29 US disclosed