SCHEMBL10679579

SCHEMBL10679579

CC1CC1n1cc(C(=O)O)c(=O)c2cc(F)c(N3CCC(N)C3)c(F)c21

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.66
POLB P06746 1/20 0.66
CHRM2 P08172 1/20 0.66
CHRM1 P11229 1/20 0.66
OPRM1 P35372 1/20 0.66
OPRD1 P41143 1/20 0.66
PIM1 P11309 1/20 0.56
GSK3A P49840 1/20 0.56
GSK3B P49841 1/20 0.56
PIM3 Q86V86 1/20 0.56
CSNK1G1 Q9HCP0 1/20 0.56
TOP2A P11388 12/20 0.55
TOP2B Q02880 10/20 0.55
TOP1 P11387 4/20 0.53
KCNH2 Q12809 1/20 0.53
LMNA P02545 1/20 0.52
KDM4E B2RXH2 1/20 0.52
HPGD P15428 1/20 0.52
HSD17B10 Q99714 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9416082 0.89 ALDH1A1 (0.82) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9416068 0.89 ALDH1A1 (0.82) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL1387312 0.89 ALDH1A1 (0.82) ALDH1A1POLBCHRM2CHRM1OPRM1
Hydrochloric Acid SCHEMBL9416083 0.88 ALDH1A1 (0.80) ALDH1A1POLBCHRM2CHRM1OPRM1
Hydrochloric Acid SCHEMBL8566510 0.88 ALDH1A1 (0.80) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL13483596 0.84 ALDH1A1 (0.82) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL10677875 0.84 KCNH2 (0.53) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9790131 0.83 ALDH1A1 (0.73) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL30626307 0.83 LMNA (0.58) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9790188 0.83 ALDH1A1 (0.73) ALDH1A1POLBCHRM2CHRM1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4777175-A (NAPHTHYRIDINE, QUINOLINE) CARBOXYLIC ACID WARNER-LAMBERT COMPANY (US) 1988-10-11 US disclosed
US-4771054-A QUINOLINE CARBOXYLIC ACID WARNER-LAMBERT COMPANY (US) 1988-09-13 US disclosed
US-4665079-A QUINOLINE DERIVATIVES WARNER-LAMBERT COMPANY (US) 1987-05-12 US disclosed
US-4638067-A NAPHTHYRIDINE AND QUINOLINE CARBOXYLIC ACIDS WARNER-LAMBERT CO. (US) 1987-01-20 US disclosed
EP-0153163-A2 7-Substituted-1-cyclopropyl-6,8-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids; 7-substituted-1-cyclopropyl-1,4-dihydro-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acids; their derivatives; and a process for preparing the compounds WARNER-LAMBERT COMPANY (US) 1985-08-28 EP disclosed