SCHEMBL10686133

SCHEMBL10686133

COc1ccc(C(C)(C)C(C)(C)c2ccc(OC)cc2F)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.49
CYP11B1 P15538 2/20 0.44
CYP11B2 P19099 2/20 0.44
CYP1A2 P05177 2/20 0.43
CYP1A1 P04798 1/20 0.43
CYP1B1 Q16678 1/20 0.43
CPS1 P31327 3/20 0.41
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
CYP2A6 P11509 1/20 0.39
AMY1A P0DUB6 3/20 0.39
TAAR1 Q96RJ0 1/20 0.38
GAA P10253 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1506600 0.88 KIF11 (0.49) KIF11CYP11B1CYP11B2CYP1A2CYP1A1
SCHEMBL531512 0.84 KIF11 (0.47) KIF11CYP11B1CYP11B2CYP1A2CYP1A1
SCHEMBL15305003 0.83 CYP11B2 (0.59) KIF11CYP11B1CYP11B2CYP1A2CYP1A1
SCHEMBL19987450 0.82 KIF11 (0.49) KIF11CYP11B1CYP11B2CYP1A2CYP1A1
SCHEMBL28661528 0.82 KIF11 (0.48) KIF11CYP11B1CYP11B2CYP1A2CYP1A1
SCHEMBL19987447 0.81 KIF11 (0.48) KIF11CYP11B1CYP11B2CYP1A2CYP1A1
SCHEMBL3993767 0.80 KIF11 (0.43) KIF11CYP11B1CYP11B2CYP1A2CYP1A1
SCHEMBL19469679 0.78 AKR1C3 (0.50) KIF11CPS1CA1CA2
Hydrochloric Acid SCHEMBL8507684 0.78 KIF11 (0.52) KIF11CYP11B1CYP11B2CYP1A2CYP1A1
SCHEMBL5187849 0.78 KIF11 (0.52) KIF11CYP11B1CYP11B2CYP1A2CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0206021-B1 DERIVATIVES OF 1,1,2,2-TETRAMETHYL-1,2-BIS(2-FLUORO-4-HYDROXYPHENYL) ETHANE ASTA Pharma AG (DE) 1988-08-10 EP disclosed
US-4745233-A Derivatives of 1,1,2,2-tetramethyl-1,2-bis-(2-fluoro-4-hydroxyphenyl)-ethane ASTA-WERKE AKTIENGESELLSCHAFT (DE) 1988-05-17 US disclosed
EP-0206021-A1 Derivatives of 1,1,2,2-tetramethyl-1,2-bis(2-fluoro-4-hydroxyphenyl) ethane ASTA Pharma AG (DE) 1986-12-30 EP disclosed