SCHEMBL10686208

SCHEMBL10686208

CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CC(C)C(CN)C3)c(F)c21

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.66
HSD17B10 Q99714 4/20 0.66
ALDH1A1 P00352 3/20 0.66
HPGD P15428 3/20 0.66
PMP22 Q01453 1/20 0.65
KCNH2 Q12809 3/20 0.45
DRD3 P35462 1/20 0.45
LMNA P02545 2/20 0.44
BRD4 O60885 1/20 0.44
TSHR P16473 1/20 0.44
HTT P42858 1/20 0.44
CYP2J2 P51589 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TOP1 P11387 3/20 0.44
CYP2C9 P11712 1/20 0.43
ATP6V1B2 P21281 1/20 0.43
TBXA2R P21731 1/20 0.43
EDNRA P25101 1/20 0.43
TARBP2 Q15633 1/20 0.43
AADAT Q8N5Z0 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10689802 0.92 KDM4E (0.67) KDM4EHSD17B10ALDH1A1HPGDPMP22
SCHEMBL10689144 0.88 KDM4E (0.68) KDM4EHSD17B10ALDH1A1HPGDPMP22
SCHEMBL10689137 0.88 KDM4E (0.68) KDM4EHSD17B10ALDH1A1HPGDPMP22
SCHEMBL10689149 0.88 KDM4E (0.68) KDM4EHSD17B10ALDH1A1HPGDPMP22
SCHEMBL10375286 0.86 KCNH2 (0.59) KDM4EHSD17B10ALDH1A1HPGDKCNH2
SCHEMBL20850987 0.83 KDM4E (0.47) KDM4EHSD17B10ALDH1A1HPGDPMP22
SCHEMBL9524138 0.83 KDM4E (0.72) KDM4EHSD17B10ALDH1A1HPGDPMP22
SCHEMBL9070334 0.83 KDM4E (0.69) KDM4EHSD17B10ALDH1A1HPGDPMP22
SCHEMBL10690023 0.83 DRD3 (0.64) KDM4EHSD17B10ALDH1A1HPGDDRD3
SCHEMBL10621416 0.82 KDM4E (0.68) KDM4EHSD17B10ALDH1A1HPGDPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4753953-A Pyridonecarboxylic acid derivatives and antibacterial pharmaceutical compositions thereof KYORIN PHARMACEUTICAL CO., LTD. (JP) 1988-06-28 US disclosed
EP-0208210-A1 Pyridonecarboxylic acid derivatives and process for their preparation KYORIN PHARMACEUTICAL CO., LTD. (JP) 1987-01-14 EP disclosed