SCHEMBL10686288

SCHEMBL10686288

NCCCS(=O)(=O)c1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.52
KMT2A Q03164 4/20 0.49
MEN1 O00255 2/20 0.49
ALDH1A1 P00352 5/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
CA2 P00918 4/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA3 P07451 1/20 0.48
CA4 P22748 1/20 0.48
CA6 P23280 1/20 0.48
CA5A P35218 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA13 Q8N1Q1 1/20 0.48
CA14 Q9ULX7 1/20 0.48
CA5B Q9Y2D0 1/20 0.48
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5708672 0.92 NPC1 (0.49) NPC1KMT2AMEN1ALDH1A1CYP3A4
SCHEMBL1939594 0.88 NPC1 (0.55) NPC1KMT2AMEN1ALDH1A1CYP3A4
SCHEMBL7413114 0.82 ALDH1A1 (0.50) NPC1KMT2AMEN1ALDH1A1CYP3A4
Hydrochloric Acid SCHEMBL7012167 0.81 F10 (0.43) ALDH1A1
SCHEMBL10724186 0.80 ALDH1A1 (0.48) NPC1KMT2AMEN1ALDH1A1CYP3A4
SCHEMBL18225990 0.80 ALDH1A1 (0.48) KMT2AMEN1ALDH1A1CYP3A4CYP2C9
SCHEMBL10568403 0.80 ALDH1A1 (0.48) NPC1KMT2AMEN1ALDH1A1CYP3A4
SCHEMBL4741649 0.80 ALDH1A1 (0.48) NPC1KMT2AMEN1ALDH1A1CYP3A4
SCHEMBL14846541 0.79 MEN1 (0.45) KMT2AMEN1ALDH1A1CYP3A4CYP2C9
SCHEMBL4409970 0.79 PSIP1 (0.52) KMT2AMEN1ALDH1A1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4724235-A N-(arylthioalkyl)-N'-(aminoalkyl)ureas useful in the treatment of arrhythmia A. H. ROBINS COMPANY, INCORPORATED (US) 1988-02-09 US disclosed
US-4597902-A TREATMENT OF CARDIAC ARRHYTHMIAS A. H. ROBINS COMPANY, INCORPORATED (US) 1986-07-01 US disclosed
EP-0066415-B1 N-(ARYLTHIOALKYL)-N'-(AMINOALKYL)UREAS A.H. ROBINS COMPANY, INCORPORATED (US) 1985-10-02 EP disclosed
EP-0066415-A2 N-(arylthioalkyl)-N'-(aminoalkyl)ureas A.H. ROBINS COMPANY, INCORPORATED (US) 1982-12-08 EP disclosed