SCHEMBL10688024

SCHEMBL10688024

CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3C[C@@H](N)[C@@H](C)C3)cc21

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 1/20 0.67
HSD17B10 Q99714 4/20 0.66
ALDH1A1 P00352 5/20 0.66
KDM4E B2RXH2 5/20 0.66
HPGD P15428 4/20 0.66
HTT P42858 3/20 0.66
LMNA P02545 2/20 0.66
TSHR P16473 2/20 0.66
BRD4 O60885 1/20 0.66
CYP2J2 P51589 1/20 0.66
NPSR1 Q6W5P4 1/20 0.66
MEN1 O00255 7/20 0.61
KMT2A Q03164 7/20 0.61
NPC1 O15118 1/20 0.61
HIF1A Q16665 1/20 0.58
USP2 O75604 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
GAA P10253 3/20 0.56
PIK3CD O00329 2/20 0.56
PIK3R1 P27986 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10688019 1.00 DRD3 (0.67) DRD3HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL10688010 1.00 DRD3 (0.67) DRD3HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL10690023 0.88 DRD3 (0.64) DRD3HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL9142833 0.85 DRD3 (0.62) DRD3HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL9142819 0.85 DRD3 (0.62) DRD3HSD17B10ALDH1A1KDM4EHPGD
Hydrochloric Acid SCHEMBL10879015 0.85 KDM4E (0.70) DRD3HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL9142824 0.85 DRD3 (0.62) DRD3HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL10685715 0.84 KDM4E (0.66) HSD17B10ALDH1A1KDM4EHPGDHTT
SCHEMBL9048236 0.84 TOP1 (0.71) DRD3HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL10685722 0.84 KDM4E (0.66) HSD17B10ALDH1A1KDM4EHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4753953-A Pyridonecarboxylic acid derivatives and antibacterial pharmaceutical compositions thereof KYORIN PHARMACEUTICAL CO., LTD. (JP) 1988-06-28 US disclosed