SCHEMBL9048236

SCHEMBL9048236

CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCC(N)C3)cc21

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 3/20 0.71
DRD3 P35462 1/20 0.70
ALDH1A1 P00352 6/20 0.68
KDM4E B2RXH2 5/20 0.68
HPGD P15428 5/20 0.68
HSD17B10 Q99714 4/20 0.68
HTT P42858 3/20 0.68
LMNA P02545 3/20 0.68
TSHR P16473 2/20 0.68
BRD4 O60885 1/20 0.68
CYP2J2 P51589 1/20 0.68
NPSR1 Q6W5P4 1/20 0.68
MEN1 O00255 7/20 0.64
KMT2A Q03164 7/20 0.64
NPC1 O15118 1/20 0.64
HIF1A Q16665 1/20 0.60
USP2 O75604 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
GAA P10253 3/20 0.59
RAD52 P43351 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8571733 0.99 TOP1 (0.70) TOP1DRD3ALDH1A1KDM4EHPGD
SCHEMBL9045019 0.90 TOP1 (0.71) TOP1DRD3ALDH1A1KDM4EHPGD
SCHEMBL10621421 0.88 TOP1 (0.72) TOP1DRD3ALDH1A1KDM4EHPGD
Hydrochloric Acid SCHEMBL8134989 0.87 TOP1 (0.56) TOP1DRD3ALDH1A1KDM4EHPGD
SCHEMBL9750328 0.86 KDM4E (0.72) TOP1DRD3ALDH1A1KDM4EHPGD
SCHEMBL9749182 0.85 DRD3 (0.69) DRD3ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL10619341 0.85 DRD3 (0.66) TOP1DRD3ALDH1A1KDM4EHPGD
SCHEMBL10620925 0.85 DRD3 (0.65) TOP1DRD3ALDH1A1KDM4EHPGD
SCHEMBL2858227 0.84 DRD3 (0.70) DRD3ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL11022977 0.84 DRD3 (0.83) DRD3ALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0360258-B1 Amino acid quinoline and naphthyridine derivatives ABBOTT LAB (US) 1996-08-14 EP disclosed
US-5057523-A Water soluble bactericide ABBOTT LABORATORIES (US) 1991-10-15 US disclosed
US-5057520-A Water solubility ABBOTT LABORATORIES (US) 1991-10-15 US disclosed
EP-0360258-A2 Amino acid quinoline and naphthyridine derivatives ABBOTT LABORATORIES (US) 1990-03-28 EP disclosed
US-4762845-A BACTERICIDES ABBOTT LABORATORIES (US) 1988-08-09 US disclosed