SCHEMBL10690051

SCHEMBL10690051

c1cc2c(c(C3CO3)c1)OCC2

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.46
HTR1A P08908 3/20 0.41
SLC6A2 P23975 3/20 0.36
SLC6A4 P31645 3/20 0.36
HRH1 P35367 1/20 0.36
SLC6A3 Q01959 1/20 0.36
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
TSHR P16473 1/20 0.33
KCNH2 Q12809 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747214 0.79 HTR1A (0.51) PARP1HTR1AADRA1A
SCHEMBL614437 0.73 HTR1A (0.46) PARP1HTR1ASLC6A2SLC6A4HRH1
SCHEMBL6677547 0.71 HTR2C (0.50) PARP1SLC6A2SLC6A4SLC6A3
SCHEMBL6677544 0.71 HTR2C (0.50) PARP1SLC6A2SLC6A4SLC6A3
SCHEMBL19699408 0.70 SLC9A1 (0.46)
SCHEMBL19690310 0.70 SLC9A1 (0.46)
SCHEMBL23323106 0.70 CHRM5 (0.44) PARP1HTR1A
SCHEMBL6677846 0.70 PARP1 (0.43) PARP1HTR1ASLC6A2SLC6A4HRH1
SCHEMBL6677848 0.70 PARP1 (0.43) PARP1HTR1ASLC6A2SLC6A4HRH1
SCHEMBL8912822 0.68 TAAR1 (0.56) SLC6A2SLC6A4HRH1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4751222-A 2,3,4,5-tetrahydro-1H-3-benzazepines and CNS affecting use thereof NOVO INDUSTRI A/S (DK) 1988-06-14 US disclosed
EP-0200455-A2 2,3,4,5-tetrahydro-1H-3-benzazepines substituted in position 5 NOVO NORDISK A/S (DK) 1986-11-05 EP disclosed