SCHEMBL10690326

SCHEMBL10690326

COc1ccc(OCc2ccccc2)c(-c2nc3nc(OC)ncc3[nH]2)c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.48
PDE4B Q07343 2/20 0.48
PDE4C Q08493 2/20 0.48
PDE4D Q08499 2/20 0.48
PDE5A O76074 1/20 0.48
PDE2A O00408 1/20 0.43
PRMT5 O14744 10/20 0.42
CYP2E1 P05181 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2B6 P20813 1/20 0.41
CYP2C19 P33261 1/20 0.41
PDGFRB P09619 1/20 0.41
PDGFRA P16234 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10691950 0.86 PDE2A (0.45) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL10691792 0.85 PDE2A (0.56) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL10685936 0.85 PDE2A (0.51) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL10689020 0.84 PDE5A (0.46) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL10690322 0.83 PDGFRB (0.43) PDE4APDE4BPDE4CPDE4DCYP2E1
SCHEMBL10692327 0.83 PDE5A (0.43) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL10611572 0.81 PDE2A (0.51) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL10690580 0.79 PDE2A (0.64) PDE5APDE2ACYP2E1CYP3A4CYP2C8
Water SCHEMBL10868986 0.78 PDE2A (0.47) PDE5APDE2APDGFRBPDGFRA
Water SCHEMBL10869421 0.78 PDE2A (0.47) PDE5APDE2APDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4722929-A Novel 2-phenyl-imidazoles and pharmaceutical compositions containing same DR. KARL THOMAE GMBH (DE) 1988-02-02 US disclosed
EP-0149200-A1 Novel 2-pnenyl-imidazoles, their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1985-07-24 EP disclosed