SCHEMBL10692327

SCHEMBL10692327

CCOc1cc(OCc2ccccc2)ccc1-c1nc2nc(OC)ncc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.43
PDE2A O00408 1/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
PRMT5 O14744 13/20 0.43
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
PDGFRB P09619 1/20 0.41
PDGFRA P16234 1/20 0.41
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40
GABRA2 P47869 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10685936 0.93 PDE2A (0.51) PDE5APDE2APDE4APDE4BPDE4C
SCHEMBL10611572 0.89 PDE2A (0.51) PDE5APDE2APDE4APDE4BPDE4C
SCHEMBL10686656 0.88 PDE2A (0.53) PDE5APDE2APDE4APDE4BPDE4C
SCHEMBL10691792 0.85 PDE2A (0.56) PDE5APDE2APDE4APDE4BPDE4C
SCHEMBL10692316 0.84 PDGFRB (0.43) PRMT5KDM4EMAPTPDGFRBPDGFRA
SCHEMBL10690326 0.83 PDE4A (0.48) PDE5APDE2APDE4APDE4BPDE4C
SCHEMBL10688934 0.82 PDE5A (0.43) PDE5APDE2APDE4APDE4BPDE4C
SCHEMBL10686094 0.82 PDE2A (0.50) PDE5APDE2APDE4APDE4BPDE4C
SCHEMBL10610931 0.81 PDE2A (0.42) PDE5APDE2APDE4APDE4BPDE4C
SCHEMBL10691950 0.79 PDE2A (0.45) PDE5APDE2APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4722929-A Novel 2-phenyl-imidazoles and pharmaceutical compositions containing same DR. KARL THOMAE GMBH (DE) 1988-02-02 US disclosed
EP-0149200-A1 Novel 2-pnenyl-imidazoles, their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1985-07-24 EP disclosed