SCHEMBL1069042

SCHEMBL1069042

O=C(CN1CCc2cc(-n3ccoc3=O)ccc2C1)N1CCN(C2CCC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 5/20 0.39
SIGMAR1 Q99720 5/20 0.39
PARP1 P09874 1/20 0.38
HRH3 Q9Y5N1 8/20 0.37
HTR1A P08908 2/20 0.37
HRH2 P25021 2/20 0.37
HRH1 P35367 2/20 0.37
CHRM4 P08173 1/20 0.37
CHRM5 P08912 1/20 0.37
ADRA2A P08913 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA1D P25100 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
DRD3 P35462 1/20 0.37
HTR2B P41595 1/20 0.37
HTR5A P47898 1/20 0.37
ALDH1A1 P00352 5/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1020589 0.82 PARP1 (0.41) TMEM97SIGMAR1PARP1HRH3HTR1A
SCHEMBL1017152 0.81 HRH3 (0.51) TMEM97SIGMAR1PARP1HRH3HTR1A
SCHEMBL1017103 0.81 HRH3 (0.49) TMEM97SIGMAR1PARP1HRH3HTR1A
SCHEMBL1016821 0.80 ALDH1A1 (0.45) TMEM97SIGMAR1PARP1HRH3CHRM4
SCHEMBL1014992 0.80 TMEM97 (0.42) TMEM97SIGMAR1PARP1HRH3HTR1A
SCHEMBL1014022 0.79 HRH3 (0.48) TMEM97SIGMAR1PARP1HRH3HTR1A
SCHEMBL1018277 0.79 TMEM97 (0.40) TMEM97SIGMAR1PARP1HRH3HTR1A
SCHEMBL1017287 0.78 FAAH (0.44) PARP1HRH3ALDH1A1PKMGAA
SCHEMBL1018373 0.78 TMEM97 (0.40) TMEM97SIGMAR1PARP1HRH3HTR1A
SCHEMBL1018194 0.78 ALDH1A1 (0.45) PARP1HRH3ALDH1A1PKMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1998620-B1 PIPERAZINYL OXOALKYL TETRAHYDROISOQUINOLINES AND RELATED ANALOGUES NEUROGEN CORP (US) 2011-01-12 EP disclosed