SCHEMBL10691491

SCHEMBL10691491

COc1ccc(C2(c3ccc(N(C)C)cc3N(C)C)OC(=O)c3cc(N(C)C)ccc32)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.67
ALDH1A1 P00352 3/20 0.67
HSD17B10 Q99714 2/20 0.67
TDP1 Q9NUW8 2/20 0.67
HPGD P15428 1/20 0.67
HIF1A Q16665 1/20 0.67
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
EDNRB P24530 1/20 0.37
EDNRA P25101 1/20 0.37
MAOB P27338 2/20 0.37
MAOA P21397 1/20 0.37
MAPT P10636 3/20 0.36
LMNA P02545 2/20 0.36
USP2 O75604 1/20 0.36
HTT P42858 1/20 0.36
CES1 P23141 1/20 0.35
GSTP1 P09211 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRL1 P41146 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9481735 0.90 ALDH1A1 (0.82) CYP3A4ALDH1A1HSD17B10TDP1HPGD
SCHEMBL10689289 0.90 ALDH1A1 (0.82) CYP3A4ALDH1A1HSD17B10TDP1HPGD
SCHEMBL10692980 0.86 CYP3A4 (0.54) CYP3A4ALDH1A1HSD17B10TDP1HPGD
SCHEMBL10692785 0.85 CYP3A4 (0.69) CYP3A4ALDH1A1HSD17B10TDP1HPGD
SCHEMBL5670276 0.84 CYP3A4 (0.75) CYP3A4ALDH1A1HSD17B10TDP1HPGD
SCHEMBL10693003 0.84 ALDH1A1 (0.67) CYP3A4ALDH1A1HSD17B10TDP1HPGD
SCHEMBL10935899 0.83 TDP1 (0.69) CYP3A4ALDH1A1HSD17B10TDP1HPGD
SCHEMBL27188 0.81 ALDH1A1 (1.00) CYP3A4ALDH1A1HSD17B10TDP1HPGD
SCHEMBL18143522 0.81 ALDH1A1 (1.00) CYP3A4ALDH1A1HSD17B10TDP1HPGD
SCHEMBL10858937 0.81 ALDH1A1 (0.65) CYP3A4ALDH1A1HSD17B10TDP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4732991-A Substituted phthalides HILTON DAVIS CHEMICAL CO. (US) 1988-03-22 US claimed
US-4732991-A Substituted phthalides HILTON DAVIS CHEMICAL CO. (US) 1988-03-22 US disclosed
US-4595768-A 3-(substituted phenyl)phthalides THE HILTON-DAVIS CHEMICAL CO. (US) 1986-06-17 US disclosed