SCHEMBL10692529

SCHEMBL10692529

COC(=O)c1ccc2cc(C(O)(c3ccccc3)c3cccnc3)ccc2c1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 10/20 0.58
CYP11B1 P15538 1/20 0.58
CYP11B2 P19099 1/20 0.58
ALDH1A1 P00352 1/20 0.51
CYP3A4 P08684 5/20 0.50
CYP17A1 P05093 1/20 0.50
CYP3A5 P20815 3/20 0.48
ACSS2 Q9NR19 1/20 0.47
ALOX15 P16050 1/20 0.45
HTT P42858 1/20 0.45
RORC P51449 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804331 0.87 CYP3A4 (0.51) CYP19A1CYP3A4CYP17A1CYP3A5RORC
SCHEMBL10690806 0.86 CYP19A1 (0.60) CYP19A1CYP11B1CYP11B2ALDH1A1CYP3A4
SCHEMBL9804417 0.77 CYP19A1 (0.55) CYP19A1CYP11B1CYP11B2CYP3A4CYP3A5
SCHEMBL13865455 0.76 TSHR (0.64) ALDH1A1ACSS2
SCHEMBL4558274 0.76 CYP19A1 (0.65) CYP19A1CYP3A4CYP3A5RORC
SCHEMBL10692778 0.75 CYP19A1 (0.69) CYP19A1CYP11B1CYP11B2ALDH1A1CYP3A4
SCHEMBL4509922 0.74 CYP11B2 (1.00) CYP19A1CYP11B1CYP11B2ALDH1A1CYP17A1
SCHEMBL913686 0.73 CYP19A1 (0.72) CYP19A1CYP3A4CYP3A5RORC
SCHEMBL10686317 0.73 CYP19A1 (0.66) CYP19A1CYP11B1CYP11B2ALDH1A1CYP3A4
SCHEMBL1519827 0.72 CYP11B1 (0.65) CYP19A1CYP11B1CYP11B2ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4734406-A 3-pyridylmethylnaphthyl derivatives and composition containing them useful to inhibit thromboxane synthetase HOECHST AKTIENGESELLSCHAFT (DE) 1988-03-29 US disclosed