SCHEMBL10693072

SCHEMBL10693072

COc1nc(C(=O)O)c(OC)c2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.46
ALDH1A1 P00352 4/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2C19 P33261 1/20 0.46
KDM4E B2RXH2 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
MAPK1 P28482 1/20 0.45
ALOX15 P16050 1/20 0.43
CYP2C9 P11712 1/20 0.41
IDO1 P14902 1/20 0.41
CDK9 P50750 1/20 0.41
DYRK1A Q13627 1/20 0.41
MAPT P10636 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
USP2 O75604 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TACR3 P29371 1/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8789401 0.79 POLB (0.44) POLBALDH1A1KDM4ESMN1; SMN2MAPK1
SCHEMBL15022582 0.77 ALOX15 (0.41) POLBALDH1A1CYP1A2KDM4ESMN1; SMN2
SCHEMBL27341760 0.76 CYP1A2 (0.64) POLBALDH1A1CYP1A2CYP2C19KDM4E
SCHEMBL4351790 0.75 POLB (0.53) POLBALDH1A1KDM4ESMN1; SMN2MAPK1
SCHEMBL31109181 0.73 SMN1; SMN2 (0.52) POLBALDH1A1CYP1A2CYP2C19SMN1; SMN2
SCHEMBL28674515 0.73 PLK1 (0.44) POLBALDH1A1CYP1A2CYP2C19KDM4E
SCHEMBL31109177 0.73 SMN1; SMN2 (0.52) POLBALDH1A1CYP1A2CYP2C19SMN1; SMN2
SCHEMBL27693524 0.72 KMT2A (0.54) POLBALDH1A1CYP2C19KDM4EALOX15
SCHEMBL394571 0.72 POLB (0.58) POLBALDH1A1KDM4EALOX15MAPT
SCHEMBL5717618 0.72 ALDH1A1 (0.67) POLBALDH1A1KDM4ESMN1; SMN2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0259838-A2 Pharmaceutical composition containing A 1,4-dihydropyridine derivative and an acylated 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid SYNTEX (U.S.A.) INC. (US) 1988-03-16 EP disclosed