SCHEMBL10693338

SCHEMBL10693338

Cc1cccc2c(C#N)csc12

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
CYP2A6 P11509 3/20 0.39
CYP1A2 P05177 2/20 0.38
AR P10275 3/20 0.36
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
PDE10A Q9Y233 1/20 0.34
IMPDH2 P12268 3/20 0.33
GRM5 P41594 2/20 0.33
IMPDH1 P20839 2/20 0.33
DYRK1A Q13627 3/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10691179 0.81 GPR35 (0.39) CYP2A6CYP1A2ALDH1A1GRM5
SCHEMBL30350331 0.78 CYP2A6 (0.39) CYP2A6ARALDH1A1KDM4EGAA
SCHEMBL29153598 0.78 CYP2A6 (0.39) CYP2A6ARALDH1A1KDM4EGAA
SCHEMBL31358012 0.78 TSHR (0.45) TSHRCYP2A6CYP1A2ARALDH1A1
SCHEMBL29915143 0.78 DYRK1A (0.46) CYP2A6ALDH1A1KDM4EGAAMAPT
SCHEMBL27002564 0.78 DYRK1A (0.46) CYP2A6ALDH1A1KDM4EGAAMAPT
SCHEMBL8404365 0.76 CYP1A2 (0.48) TSHRCYP2A6CYP1A2ALDH1A1GAA
SCHEMBL10692886 0.75 PTGS1 (0.38) CYP2A6CYP1A2KDM4E
SCHEMBL10693094 0.75 IFNAR1 (0.44) TSHRCYP2A6ALDH1A1KDM4EGAA
SCHEMBL10692882 0.75 PTGS1 (0.38) CYP2A6CYP1A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117500799-A Substituted fused azines as KRAS G12D inhibitors 伊莱利利公司 2024-02-02 CN disclosed
US-4737516-A FUNGICIDES SANDOZ LTD. (CH) 1988-04-12 US disclosed