SCHEMBL10693428

SCHEMBL10693428

COC(=O)C([C@@H](C)O[Si](C)(C)C(C)(C)C)N1C(=O)C(N2C(=O)c3ccccc3C2=O)C1C(O)C(=O)c1ccc(Cl)cc1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 3/20 0.34
TP53 P04637 2/20 0.34
NPSR1 Q6W5P4 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KMT2A Q03164 3/20 0.32
ALDH1A1 P00352 2/20 0.32
NPC1 O15118 1/20 0.32
CYP1A2 P05177 1/20 0.32
GAA P10253 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
RAB9A P51151 1/20 0.32
RECQL P46063 1/20 0.32
AVPR1A P37288 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694864 0.90 AVPR1A (0.42) MDM2TP53RECQLAVPR1A
SCHEMBL9228271 0.84 KMT2A (0.36) MDM2TP53NPSR1L3MBTL1KMT2A
SCHEMBL9228267 0.84 KMT2A (0.36) MDM2TP53NPSR1L3MBTL1KMT2A
SCHEMBL9222237 0.75 AVPR1A (0.39) MDM2TP53KMT2AALDH1A1NPC1
SCHEMBL9222234 0.75 AVPR1A (0.39) MDM2TP53KMT2AALDH1A1NPC1
SCHEMBL9219312 0.70 AVPR1A (0.44) CYP2D6CYP2C9CYP2C19RAB9AAVPR1A
SCHEMBL9219306 0.70 AVPR1A (0.44) CYP2D6CYP2C9CYP2C19RAB9AAVPR1A
SCHEMBL22672484 0.64 TSHR (0.34) L3MBTL1KMT2AALDH1A1GAACYP2C19
SCHEMBL24064546 0.63 TSHR (0.35) L3MBTL1KMT2AALDH1A1GAACYP2C19
SCHEMBL10670704 0.63 TP53 (0.39) TP53NPSR1L3MBTL1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0282895-A2 2-oxa-isocephem compounds, compositions containing same and processes for preparing same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-09-21 EP disclosed