SCHEMBL10694013

SCHEMBL10694013

CC(=O)c1ccc(OC(CCCCC(=O)O)c2ccc(-c3ccccc3)cc2)cc1O

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 1/20 0.47
MAOB P27338 5/20 0.47
SLC6A9 P48067 5/20 0.45
ALDH1A1 P00352 2/20 0.45
CYP2D6 P10635 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
SLC6A5 Q9Y345 1/20 0.45
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
MAPK1 P28482 1/20 0.42
GCGR P47871 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10691549 0.93 MAOB (0.51) PPARDMAOBALDH1A1CYP3A4HPGD
SCHEMBL10691499 0.89 MAOB (0.51) PPARDMAOB
SCHEMBL10693512 0.79 PPARD (0.52) PPARDMAOBALDH1A1CYP3A4HPGD
SCHEMBL10692952 0.78 CYSLTR2 (0.53) PPARDMAPTCYP2C9
SCHEMBL10693027 0.76 PPARD (0.49) PPARDMAOBALDH1A1CYP3A4HPGD
SCHEMBL10687936 0.72 PPARD (0.71) PPARDMAOB
SCHEMBL21052036 0.72 PPARD (0.74) PPARDMAOBALDH1A1CYP3A4HPGD
SCHEMBL10691238 0.70 CYSLTR2 (0.57) PPARDMAPTCYP2C9
SCHEMBL4216869 0.69 ACMSD (0.72) MAOBALDH1A1MAPTCYP3A4HPGD
SCHEMBL9774479 0.69 MAOB (0.58) PPARDMAOBALDH1A1CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4769482-A Cyano and thiocyano intermediates ELI LILLY AND COMPANY (US) 1988-09-06 US disclosed
EP-0108592-B1 LEUKOTRIENE ANTAGONISTS ELI LILLY AND COMPANY (US) 1987-09-30 EP disclosed
US-4661505-A 4-(4-ACETYL-3-HYDROXY-2-PROPYLPHENOXY) ALKANOIC ACIDS, TETRAZOLES, AND DERIVATIVES ELI LILLY AND COMPANY (US) 1987-04-28 US disclosed
EP-0108592-A1 Leukotriene antagonists ELI LILLY AND COMPANY (US) 1984-05-16 EP disclosed