SCHEMBL1069430

SCHEMBL1069430

COc1[c]c(OC)cc(-c2ccccc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
PDE4B Q07343 4/20 0.42
MAPT P10636 4/20 0.42
PDE4A P27815 2/20 0.42
PDE4C Q08493 2/20 0.42
PDE4D Q08499 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
TSHR P16473 1/20 0.42
ATM Q13315 1/20 0.42
CYP1A1 P04798 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2E1 P05181 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP4B1 P13584 1/20 0.41
CYP2B6 P20813 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4928847 0.88 PDE4B (0.35) ALDH1A1PDE4BMAPTPDE4APDE4C
SCHEMBL4853131 0.87 ABL1 (0.36) ALDH1A1MAPTCYP1A1CYP1A2CYP2E1
SCHEMBL455425 0.85 MAPT (0.34) ALDH1A1PDE4BMAPTPDE4APDE4C
SCHEMBL4854196 0.79 ABL1 (0.33) CYP1A1CYP1A2CYP2E1CYP3A4CYP2C8
SCHEMBL357701 0.79 CYP11B1 (0.40) ALDH1A1PDE4BMAPTPDE4APDE4C
SCHEMBL7468946 0.77 CYP11B1 (0.42) ALDH1A1PDE4BMAPTPDE4APDE4C
SCHEMBL28926451 0.77 PTPRC (0.49) ALDH1A1MAPTMEN1KMT2ATSHR
SCHEMBL28926431 0.76 ERN1 (0.47) ALDH1A1MAPTCYP1A1CYP1A2CYP1B1
SCHEMBL8617732 0.74 CA9 (0.50) ALDH1A1MAPTMEN1KMT2ATSHR
Methoxy Aucuparin SCHEMBL8420787 0.74 KDM4E (0.62) ALDH1A1MAPTMEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006886-A2 AZOLE COMPOUNDS CARRYING A SULFUR SUBSTITUENT XIV BASF SE (DE) 2011-01-20 WO disclosed
EP-1144381-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GmbH (DE) 2001-10-17 EP disclosed
EP-1133475-A1 SUBSTITUTED BENZO DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GmbH (DE) 2001-09-19 EP disclosed
WO-2000032577-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GMBH (DE) 2000-06-08 WO disclosed
WO-2000031039-A1 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GMBH (DE) 2000-06-02 WO disclosed