SCHEMBL10695543

SCHEMBL10695543

CCCCn1c(=O)n(CCC(C)=O)c(=O)c2c1ncn2CC(C)=O

nearest known ligand 0.91

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 12/20 0.91
PDE4B Q07343 11/20 0.91
PDE4C Q08493 11/20 0.91
PDE4D Q08499 11/20 0.91
ADORA2A P29274 4/20 0.91
ADORA2B P29275 3/20 0.91
LMNA P02545 2/20 0.61
CYP1A2 P05177 2/20 0.61
NFKB1 P19838 2/20 0.61
ACHE P22303 2/20 0.61
PMP22 Q01453 2/20 0.61
ESR1 P03372 1/20 0.61
MAPT P10636 1/20 0.61
BLM P54132 1/20 0.61
TRPA1 O75762 1/20 0.53
TNF P01375 2/20 0.51
RXFP1 Q9HBX9 2/20 0.51
USP2 O75604 1/20 0.51
TSHR P16473 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694108 1.00 PDE4A (0.91) PDE4APDE4BPDE4CPDE4DADORA2A
Denbufylline SCHEMBL7299526 0.95 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
Denbufylline SCHEMBL127152 0.95 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9853391 0.94 PDE4A (0.88) PDE4APDE4BPDE4CPDE4DADORA2A
Denbufylline SCHEMBL11044404 0.94 PDE4A (0.97) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10872056 0.93 PDE4A (0.95) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10696123 0.93 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7323464 0.92 PDE4A (0.93) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL11395350 0.92 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7800770 0.92 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0260127-A2 Xanthine derivatives, their preparation and pharmaceutical compositions containing them BEECHAM - WUELFING GmbH & Co. KG (DE) 1988-03-16 EP claimed
EP-0260127-A2 Xanthine derivatives, their preparation and pharmaceutical compositions containing them BEECHAM - WUELFING GmbH & Co. KG (DE) 1988-03-16 EP disclosed