SCHEMBL10695834

SCHEMBL10695834

O=C(O)C1(I)CCCN1Cc1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
HRH3 Q9Y5N1 1/20 0.40
SIGMAR1 Q99720 2/20 0.40
HSD11B1 P28845 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL288660 0.73 HTT (0.43) ALDH1A1CNR1CNR2
SCHEMBL10355477 0.70 ALDH1A1 (0.41) ALDH1A1KMT2A
SCHEMBL5067826 0.70 MEN1 (0.46) ALDH1A1SIGMAR1MEN1KMT2A
SCHEMBL11888852 0.69 ALDH1A1 (0.56) ALDH1A1HRH3MEN1KMT2A
SCHEMBL15923278 0.69 CYP2D6 (0.46) ALDH1A1MEN1KMT2A
SCHEMBL15665132 0.69 CYP2D6 (0.46) ALDH1A1MEN1KMT2A
SCHEMBL27952439 0.69 CYP2D6 (0.46) ALDH1A1MEN1KMT2A
SCHEMBL10215060 0.68 ALDH1A1 (0.43) ALDH1A1HRH3SIGMAR1HSD11B1MEN1
SCHEMBL1147459 0.68 ALDH1A1 (0.58) ALDH1A1HRH3MEN1KMT2A
SCHEMBL15664723 0.68 OPRL1 (0.45) ALDH1A1SIGMAR1HSD11B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0253785-A1 Efficient stereoconservative syntheses of 1-substituted (S)- and (R)-2-aminomethylpyrrolidines and intermediates therein ASTRA LAKEMEDEL AKTIEBOLAG (SE) 1988-01-20 EP disclosed