SCHEMBL288660

SCHEMBL288660

O=C1CCC(I)(C(=O)O)N1Cc1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.43
TSHR P16473 1/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
ALDH1A1 P00352 4/20 0.38
PTGER4 P35408 1/20 0.37
PTGER2 P43116 1/20 0.37
LMNA P02545 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MGLL Q99685 1/20 0.37
MAPT P10636 1/20 0.37
POLB P06746 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4460381 0.88 HCRTR1 (0.41) TSHRALDH1A1POLBHPGD
SCHEMBL290017 0.85 KMT2A (0.43) ALDH1A1PTGER4PTGER2SMN1; SMN2KDM4E
SCHEMBL288186 0.77 SMN1; SMN2 (0.46) HTTALDH1A1PTGER4PTGER2LMNA
SCHEMBL288848 0.75 NPSR1 (0.57) ALDH1A1PTGER4PTGER2LMNASMN1; SMN2
SCHEMBL10695834 0.73 ALDH1A1 (0.43) CNR1CNR2ALDH1A1
SCHEMBL28271896 0.71 AMPD2 (0.39) TSHRALDH1A1LMNAMAPT
SCHEMBL3733166 0.70 TSHR (0.52) TSHRALDH1A1LMNASMN1; SMN2
SCHEMBL8876707 0.66 ALDH1A1 (0.50) TSHRALDH1A1HPGD
SCHEMBL14828739 0.66 TSHR (0.51) TSHRALDH1A1LMNASMN1; SMN2
SCHEMBL14828734 0.65 ALDH1A1 (0.49) TSHRALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427429-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS Abbott GmbH & Co. KG (DE) 2012-03-14 EP disclosed
WO-2010128102-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS ABBOTT GMBH & CO. KG (DE) 2010-11-11 WO disclosed