SCHEMBL10696008

SCHEMBL10696008

CCCCn1c(=O)[nH]c2ncn(CC3(C)OCCO3)c2c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 6/20 0.46
PDE4A P27815 4/20 0.46
ADORA2A P29274 4/20 0.46
PDE4B Q07343 4/20 0.46
PDE4C Q08493 4/20 0.46
PDE4D Q08499 4/20 0.46
ADORA3 P0DMS8 3/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
ALDH1A1 P00352 2/20 0.45
CNOT7 Q9UIV1 3/20 0.44
BRD4 O60885 1/20 0.44
BRD2 P25440 1/20 0.44
BRD3 Q15059 1/20 0.44
BRDT Q58F21 1/20 0.44
RGS12 O14924 2/20 0.37
NPC1 O15118 1/20 0.37
USP2 O75604 1/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10695072 0.83 MEN1 (0.69) ADORA2BPDE4AADORA2APDE4BPDE4C
SCHEMBL11058131 0.81 PDE4A (0.62) ADORA2BPDE4AADORA2APDE4BPDE4C
SCHEMBL10696644 0.78 ADORA2B (0.65) ADORA2BPDE4AADORA2APDE4BPDE4C
SCHEMBL11054535 0.78 PDE4A (0.58) ADORA2BPDE4AADORA2APDE4BPDE4C
SCHEMBL11046863 0.77 PDE4A (0.60) ADORA2BPDE4AADORA2APDE4BPDE4C
SCHEMBL10696881 0.75 CNOT7 (0.53) ADORA2BPDE4AADORA2APDE4BPDE4C
SCHEMBL9842841 0.75 PDE4A (0.49) ADORA2BPDE4AADORA2APDE4BPDE4C
SCHEMBL10693464 0.75 PDE4A (0.63) ADORA2BPDE4AADORA2APDE4BPDE4C
SCHEMBL10694058 0.75 PDE4A (0.63) ADORA2BPDE4AADORA2APDE4BPDE4C
SCHEMBL5174205 0.73 ADORA2B (0.51) ADORA2BPDE4AADORA2APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0260127-A2 Xanthine derivatives, their preparation and pharmaceutical compositions containing them BEECHAM - WUELFING GmbH & Co. KG (DE) 1988-03-16 EP disclosed