SCHEMBL10696558

SCHEMBL10696558

COc1cc(CCNCCc2cc(OC)c(OC)c(OC)c2)cc(OC)c1OC

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.62
HTR2C P28335 1/20 0.62
HTR2B P41595 1/20 0.62
CA12 O43570 1/20 0.62
CA1 P00915 1/20 0.62
CA2 P00918 1/20 0.62
CA9 Q16790 1/20 0.62
CA14 Q9ULX7 1/20 0.62
PTGS2 P35354 1/20 0.57
TUBB4A P04350 3/20 0.56
TUBB P07437 3/20 0.56
TUBA3C P0DPH7 3/20 0.56
TUBA1B P68363 3/20 0.56
TUBA4A P68366 3/20 0.56
TUBB4B P68371 3/20 0.56
TUBB3 Q13509 3/20 0.56
TUBB2A Q13885 3/20 0.56
TUBB8 Q3ZCM7 3/20 0.56
TUBA3E Q6PEY2 3/20 0.56
TUBA1A Q71U36 3/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1677780 0.90 CA12 (0.57) HTR2AHTR2CHTR2BCA12CA1
SCHEMBL4320087 0.86 POLB (0.65) HTR2AHTR2CHTR2BCA12CA1
SCHEMBL3199504 0.85 KMT2A (0.54) HTR2AHTR2CHTR2BCA12CA1
SCHEMBL6775446 0.84 CA12 (0.51) HTR2AHTR2CHTR2BCA12CA1
SCHEMBL4464142 0.84 HTR2A (0.75) HTR2AHTR2CHTR2BCA12CA1
Hydrochloric Acid SCHEMBL9829288 0.84 POLB (0.62) HTR2AHTR2CHTR2BCA12CA1
SCHEMBL10501194 0.83 CA12 (0.58) HTR2AHTR2CHTR2BCA12CA1
SCHEMBL1967247 0.83 ALDH1A1 (0.50) HTR2AHTR2CHTR2BCA12CA1
SCHEMBL8533124 0.82 GAA (0.60) PTGS2TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8026574 0.82 GAA (0.60) PTGS2TUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0251194-A1 Use of carbocyclic and heterocyclic condensed dihydropyridines for the preparation of cardioprotective remedies and heterocyclic and carbocyclic condensed dihydropyridines and methods and intermediates for their preparation BOEHRINGER INGELHEIM KG (DE) 1988-01-07 EP claimed
EP-0251194-A1 Use of carbocyclic and heterocyclic condensed dihydropyridines for the preparation of cardioprotective remedies and heterocyclic and carbocyclic condensed dihydropyridines and methods and intermediates for their preparation BOEHRINGER INGELHEIM KG (DE) 1988-01-07 EP disclosed