SCHEMBL10696877

SCHEMBL10696877

COC(=O)CC(C)(C)C(=O)c1ccc(SC)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.45
SMN1; SMN2 Q16637 5/20 0.44
ALDH1A1 P00352 4/20 0.44
TSHR P16473 3/20 0.44
MAPK1 P28482 1/20 0.44
EPHX2 P34913 1/20 0.43
NR1H4 Q96RI1 1/20 0.43
HAO1 Q9UJM8 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
MAPT P10636 7/20 0.40
HTT P42858 3/20 0.40
GAA P10253 2/20 0.40
ALOX15 P16050 1/20 0.40
KDM4E B2RXH2 4/20 0.37
LMNA P02545 3/20 0.36
NPSR1 Q6W5P4 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10699043 0.82 CA1 (0.48) ALDH1A1TSHRMAPK1MAPTGAA
SCHEMBL6153059 0.81 KMT2A (0.48) SMN1; SMN2ALDH1A1MAPK1MAPTHTT
SCHEMBL6399385 0.81 MAPK1 (0.51) PLK1SMN1; SMN2ALDH1A1MAPK1EPHX2
SCHEMBL6400649 0.81 POLB (0.44) SMN1; SMN2ALDH1A1MAPK1MAPTKDM4E
SCHEMBL5183124 0.80 SRC (0.51) SMN1; SMN2ALDH1A1TSHRMAPK1MAPT
SCHEMBL14632299 0.79 EPHX2 (0.44) SMN1; SMN2ALDH1A1EPHX2NR1H4MAPT
SCHEMBL9733471 0.79 ALDH1A1 (0.36) PLK1SMN1; SMN2ALDH1A1MAPTGAA
SCHEMBL17295068 0.75 HAO1 (0.58) PLK1SMN1; SMN2ALDH1A1TSHRMAPK1
SCHEMBL5768900 0.75 HAO1 (0.58) PLK1SMN1; SMN2ALDH1A1TSHRMAPK1
SCHEMBL13610814 0.74 ALDH1A1 (0.56) PLK1SMN1; SMN2ALDH1A1TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0252639-A1 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1988-01-13 EP disclosed
EP-0104885-B1 LEUKOTRIENE ANTAGONISTS, THEIR PRODUCTION, AND COMPOSITIONS CONTAINING THEM MERCK FROSST CANADA INC. (CA) 1986-06-04 EP disclosed