SCHEMBL10696985

SCHEMBL10696985

Cc1cc(-c2nc3cc4c(cc3[nH]2)N(C(C)C)C(=O)C4(C)C)co1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.40
AURKB Q96GD4 2/20 0.40
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
BRD4 O60885 1/20 0.33
HPSE Q9Y251 1/20 0.31
ALDH1A1 P00352 1/20 0.31
PTGER3 P43115 1/20 0.30
GUSB P08236 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10701072 0.83 AURKA (0.59) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10698460 0.80 AURKA (0.48) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10695935 0.80 AURKA (0.48) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10698186 0.79 PDE4A (0.40) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10699199 0.78 MAPT (0.51) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL6454096 0.75 NPC1 (0.47) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL4827138 0.74 AURKA (0.40) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL5618911 0.74 AURKA (0.50) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL4886259 0.73 FGFR1 (0.48) AURKAAURKBALDH1A1
SCHEMBL4946021 0.73 AURKA (0.39) AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed