SCHEMBL10697190

SCHEMBL10697190

CCN1C(=O)C(C)(C)c2cc3nc(-c4ccc(C)c(S)c4OC)[nH]c3cc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.54
AURKB Q96GD4 3/20 0.54
AMY1A P0DUB6 8/20 0.43
CHEK1 O14757 1/20 0.38
SRC P12931 1/20 0.38
CDK2 P24941 1/20 0.38
KDR P35968 1/20 0.38
FLT3 P36888 1/20 0.38
GSK3B P49841 1/20 0.38
BRD4 O60885 1/20 0.36
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ATM Q13315 1/20 0.33
ERAP1 Q9NZ08 1/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
NPBWR1 P48145 2/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10697449 0.83 AURKA (0.57) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10697198 0.79 AURKA (0.51) AURKAAURKBAMY1ACHEK1SRC
SCHEMBL10373866 0.79 PDE4A (0.50) AURKAAURKBAMY1ANPC1RAB9A
SCHEMBL10701197 0.79 AURKA (0.57) AURKAAURKBKDRNPC1RAB9A
Hydrochloric Acid SCHEMBL10698205 0.78 AURKA (0.52) AURKAAURKBAMY1ACHEK1SRC
Hydrochloric Acid SCHEMBL10699432 0.76 AURKA (0.56) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10696432 0.76 AURKA (0.48) AURKAAURKBCHEK1SRCCDK2
SCHEMBL4957006 0.75 AURKA (0.66) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10696602 0.75 AURKA (0.60) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10700525 0.75 AURKA (0.61) AURKAAURKBCHEK1SRCCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed