SCHEMBL10696432

SCHEMBL10696432

CCCN1C(=O)C(C)(C)c2cc3nc(-c4ccc(C)cc4S)[nH]c3cc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.48
AURKB Q96GD4 3/20 0.48
NPBWR1 P48145 1/20 0.36
MAPT P10636 4/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TP53 P04637 3/20 0.34
SSTR2 P30874 1/20 0.33
KCNH2 Q12809 1/20 0.33
HPGD P15428 1/20 0.32
RECQL P46063 1/20 0.32
HSD17B10 Q99714 1/20 0.32
BRD4 O60885 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10697347 0.94 AURKA (0.46) AURKAAURKBNPBWR1MAPTKDM4E
SCHEMBL10697449 0.92 AURKA (0.57) AURKAAURKBNPBWR1MAPTKDM4E
SCHEMBL10696033 0.79 PDE4A (0.54) AURKAAURKBKDM4EALDH1A1GAA
SCHEMBL13341256 0.78 AURKA (0.49) AURKAAURKBNPBWR1MAPTKDM4E
SCHEMBL10699765 0.77 AURKA (0.48) AURKAAURKBMAPTKDM4EALDH1A1
SCHEMBL10694262 0.77 AURKB (0.48) AURKAAURKBNPBWR1BRD4PDE4A
SCHEMBL10696997 0.77 AURKA (0.48) AURKAAURKBMAPTKDM4EALDH1A1
SCHEMBL13367949 0.76 AURKA (0.47) AURKAAURKBKDM4EALDH1A1BRD4
SCHEMBL10695470 0.76 MAPT (0.49) AURKAAURKBMAPTKDM4EALDH1A1
SCHEMBL10697190 0.76 AURKA (0.54) AURKAAURKBNPBWR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed