SCHEMBL10697452

SCHEMBL10697452

CCN1C(=O)C(C)(C)c2cc3nc(-c4ccc(SC)cc4)[nH]c3cc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 3/20 0.57
AURKA O14965 2/20 0.57
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
BRD4 O60885 1/20 0.37
CHEK1 O14757 2/20 0.37
SRC P12931 1/20 0.37
CDK2 P24941 1/20 0.37
KDR P35968 1/20 0.37
FLT3 P36888 1/20 0.37
GSK3B P49841 1/20 0.37
CHEK2 O96017 1/20 0.37
NPBWR1 P48145 3/20 0.36
PRKD3 O94806 1/20 0.36
PAK4 O96013 1/20 0.36
PDGFRA P16234 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694262 0.92 AURKB (0.48) AURKBAURKAPDE4APDE4BPDE4C
SCHEMBL10695207 0.89 AURKB (0.46) AURKBAURKAPDE4APDE4BPDE4C
SCHEMBL10698143 0.87 AURKA (0.59) AURKBAURKAPDE4APDE4BPDE4C
SCHEMBL10698507 0.87 AURKB (0.59) AURKBAURKAPDE4APDE4BPDE4C
SCHEMBL10696602 0.86 AURKA (0.60) AURKBAURKAPDE4APDE4BPDE4C
SCHEMBL10699037 0.85 AURKA (0.57) AURKBAURKAPDE4APDE4BPDE4C
SCHEMBL10701197 0.85 AURKA (0.57) AURKBAURKAPDE4APDE4BPDE4C
SCHEMBL10699579 0.85 AURKA (0.57) AURKBAURKAPDE4APDE4BPDE4C
SCHEMBL10698462 0.84 AURKA (0.58) AURKBAURKANPBWR1CYP2C9CYP2C19
SCHEMBL10700799 0.84 AURKA (0.56) AURKBAURKANPBWR1NPC1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed