SCHEMBL10698507

SCHEMBL10698507

CCN1C(=O)C(C)(C)c2cc3nc(-c4ccc(O)cc4)[nH]c3cc21

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 3/20 0.59
AURKA O14965 2/20 0.59
NPBWR1 P48145 1/20 0.44
SCD O00767 1/20 0.43
GUSB P08236 1/20 0.42
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
TOP1 P11387 2/20 0.40
TOP2A P11388 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
DGAT1 O75907 1/20 0.40
KCNH2 Q12809 1/20 0.40
CHEK1 O14757 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10699139 0.89 AURKB (0.47) AURKBAURKANPBWR1SCDGUSB
SCHEMBL10698143 0.89 AURKA (0.59) AURKBAURKANPBWR1PDE4APDE4B
SCHEMBL10696602 0.88 AURKA (0.60) AURKBAURKASCDGUSBPDE4A
SCHEMBL10699037 0.87 AURKA (0.57) AURKBAURKANPBWR1GUSBPDE4A
SCHEMBL10701197 0.87 AURKA (0.57) AURKBAURKANPBWR1GUSBPDE4A
SCHEMBL10697452 0.87 AURKB (0.57) AURKBAURKANPBWR1PDE4APDE4B
SCHEMBL10699579 0.87 AURKA (0.57) AURKBAURKAPDE4APDE4BPDE4C
SCHEMBL10698967 0.87 AURKB (0.47) AURKBAURKANPBWR1SCDGUSB
SCHEMBL10700799 0.86 AURKA (0.56) AURKBAURKANPBWR1GUSBALDH1A1
SCHEMBL10696315 0.86 AURKA (0.56) AURKBAURKANPBWR1SCDGUSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed