SCHEMBL10698026

SCHEMBL10698026

CCN1C(=O)C(C)(C)c2cc3nc(-c4ccc(C)nc4)[nH]c3cc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.58
AURKB Q96GD4 2/20 0.58
NPC1 O15118 8/20 0.46
RAB9A P51151 8/20 0.46
PKM P14618 1/20 0.46
MITF O75030 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
KDM4E B2RXH2 10/20 0.39
ALDH1A1 P00352 10/20 0.39
MAPT P10636 8/20 0.39
HPGD P15428 7/20 0.39
BRD4 O60885 1/20 0.39
CHEK1 O14757 1/20 0.38
SRC P12931 1/20 0.38
CDK2 P24941 1/20 0.38
KDR P35968 1/20 0.38
FLT3 P36888 1/20 0.38
GSK3B P49841 1/20 0.38
PDE4A P27815 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10700213 0.86 AURKA (0.56) AURKAAURKBNPC1RAB9AKDM4E
SCHEMBL10699499 0.84 AURKA (0.57) AURKAAURKBNPC1RAB9AMITF
SCHEMBL10698143 0.84 AURKA (0.59) AURKAAURKBNPC1RAB9APKM
SCHEMBL10698507 0.84 AURKB (0.59) AURKAAURKBALDH1A1HPGDBRD4
SCHEMBL10696602 0.83 AURKA (0.60) AURKAAURKBNPC1RAB9AKDM4E
SCHEMBL10701197 0.82 AURKA (0.57) AURKAAURKBNPC1RAB9APKM
SCHEMBL10699037 0.82 AURKA (0.57) AURKAAURKBNPC1RAB9APKM
SCHEMBL10697452 0.82 AURKB (0.57) AURKAAURKBNPC1RAB9AALDH1A1
SCHEMBL10699579 0.82 AURKA (0.57) AURKAAURKBKDM4EALDH1A1MAPT
SCHEMBL10696315 0.82 AURKA (0.56) AURKAAURKBNPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed