SCHEMBL10698199

SCHEMBL10698199

Cn1c(-c2ccccn2)nc2cc3c(cc21)CC(=O)N3CCO

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 3/20 0.36
HSD17B10 Q99714 3/20 0.36
HRH3 Q9Y5N1 2/20 0.36
HTT P42858 1/20 0.36
BMPR1B O00238 1/20 0.36
BMPR1A P36894 1/20 0.36
TGFBR1 P36897 1/20 0.36
ACVRL1 P37023 1/20 0.36
ACVR1 Q04771 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10701670 0.90 NPC1 (0.48) CA12CA9NPC1RAB9AL3MBTL1
SCHEMBL10699776 0.86 CA12 (0.44) CA12CA9NPC1RAB9AL3MBTL1
SCHEMBL10699129 0.85 NPC1 (0.48) CA12CA9NPC1RAB9AL3MBTL1
SCHEMBL10696205 0.85 CA12 (0.51) CA12CA9NPC1RAB9AL3MBTL1
SCHEMBL10698954 0.81 CYP11B1 (0.48) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL10697210 0.81 CA12 (0.51) CA12CA9NPC1RAB9AL3MBTL1
SCHEMBL10702791 0.80 BMPR1B (0.42) CA12CA9MEN1KMT2AHDAC1
SCHEMBL10699035 0.79 CA12 (0.45) CA12CA9NPC1RAB9AL3MBTL1
SCHEMBL10698291 0.78 HDAC1 (0.42) HDAC1HDAC8KDM4EALDH1A1HSD17B10
SCHEMBL10700187 0.77 CA12 (0.45) CA12CA9NPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed