SCHEMBL10698214

SCHEMBL10698214

CN(C)CCOc1ccc(C/C=C(/Cc2ccc(OP(=O)(O)O)cc2)c2ccc(Br)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 4/20 0.40
ESRRB O95718 1/20 0.40
LTB4R Q15722 1/20 0.39
LTB4R2 Q9NPC1 1/20 0.39
HRH3 Q9Y5N1 2/20 0.39
UTS2R Q9UKP6 2/20 0.39
PPARD Q03181 1/20 0.39
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
LSS P48449 4/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
CYP2D6 P10635 1/20 0.37
LTA4H P09960 1/20 0.37
ESR1 P03372 2/20 0.36
ESR2 Q92731 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10698657 0.88 GBA1 (0.38) ESRRBHRH3DRD2DRD3KEAP1
SCHEMBL10780217 0.78 LTA4H (0.58) ESRRGESRRBHRH3DRD2DRD3
SCHEMBL7152772 0.78 LTA4H (0.58) ESRRGESRRBHRH3DRD2DRD3
SCHEMBL7807866 0.78 CYP2D6 (0.51) ESRRGESRRBDRD2DRD3BCHE
SCHEMBL11567088 0.77 ESR1 (0.50) ESRRGESRRBHRH3KEAP1NFE2L2
SCHEMBL7809033 0.77 ESR1 (0.53) ESRRGESRRBHRH3KEAP1NFE2L2
SCHEMBL11564379 0.76 ESR1 (0.49) ESRRGESRRBHRH3KEAP1NFE2L2
SCHEMBL9857672 0.76 ESR1 (0.63) ESRRGESRRBDRD2DRD3CYP2D6
SCHEMBL7809032 0.76 LTA4H (0.52) ESRRGDRD2DRD3BCHEACHE
SCHEMBL9857681 0.76 ESR1 (0.63) ESRRGESRRBDRD2DRD3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0272330-A1 1,1,2-TRIARYL-1-BUTENE DERIVATIVES TAIHO PHARMACEUTICAL COMPANY LIMITED (JP) 1988-06-29 EP disclosed