SCHEMBL1070286

SCHEMBL1070286

CCOC(=O)C=C(c1ccccc1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
NPC1 O15118 2/20 0.53
MAPT P10636 5/20 0.53
ALDH1A1 P00352 2/20 0.49
LMNA P02545 2/20 0.47
MDM4 O15151 1/20 0.47
MDM2 Q00987 1/20 0.47
GAA P10253 3/20 0.46
PIN1 Q13526 1/20 0.46
PTGS2 P35354 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8999208 0.93 NPC1 (0.50) MEN1KMT2ANPC1MAPTALDH1A1
SCHEMBL8999201 0.93 NPC1 (0.50) MEN1KMT2ANPC1MAPTALDH1A1
SCHEMBL6338797 0.92 L3MBTL1 (0.50) MEN1KMT2ANPC1MAPTALDH1A1
SCHEMBL5500811 0.92 L3MBTL1 (0.50) MEN1KMT2ANPC1MAPTALDH1A1
SCHEMBL5500812 0.92 L3MBTL1 (0.50) MEN1KMT2ANPC1MAPTALDH1A1
SCHEMBL433413 0.92 ESR1 (0.53) MEN1KMT2ANPC1MAPTALDH1A1
SCHEMBL433415 0.92 ESR1 (0.53) MEN1KMT2ANPC1MAPTALDH1A1
SCHEMBL1744974 0.91 NPC1 (0.48) MEN1KMT2ANPC1MAPTALDH1A1
SCHEMBL1744978 0.91 NPC1 (0.48) MEN1KMT2ANPC1MAPTALDH1A1
SCHEMBL1744976 0.91 NPC1 (0.48) MEN1KMT2ANPC1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 88 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10953256-B2 Composition comprising fluorine-containing ketone SINOCHEM LANTIAN CO., LTD (CN) 2021-03-23 US claimed
EP-3421105-A1 COMPOSITION COMPRISING FLUORINE-CONTAINING KETONE Sinochem Lantian Co., Ltd. (CN) 2019-01-02 EP claimed
US-20180200553-A1 COMPOSITION COMPRISING FLUORINE-CONTAINING KETONE SINOCHEM LANTIAN CO., LTD (CN) 2018-07-19 US claimed
WO-2022255228-A1 COMPOSITION, CURED PRODUCT OR COMPACT, OPTICAL MEMBER, AND LENS 富士フイルム株式会社 2022-12-08 WO disclosed
US-11485725-B2 Derivatives of piperlongumine and uses thereof AURANSA INC. (US) 2022-11-01 US disclosed
CN-113233980-B Synthesis method of beta-chloroacid ester and alpha, beta-unsaturated acid ester compound 台州学院 2022-04-05 CN disclosed
EP-3886633-A1 CUSHIONING ELEMENT UTILIZING FOAM PARTICLES NIKE Innovate C.V. (US) 2021-10-06 EP disclosed
CN-113233980-A Synthesis method of beta-chloroacid ester and alpha, beta-unsaturated acid ester compound 台州学院 2021-08-10 CN disclosed
US-20210198235-A1 DERIVATIVES OF PIPERLONGUMINE AND USES THEREOF AURANSA INC. 2021-07-01 US disclosed
US-20210198235-A1 DERIVATIVES OF PIPERLONGUMINE AND USES THEREOF AURANSA INC. 2021-07-01 US disclosed
EP-3836816-A1 FOOTWEAR SOLE STRUCTURE HAVING A COMPOSITE ELEMENT AND METHODS FOR MANUFACTURING SAME NIKE Innovate C.V. (US) 2021-06-23 EP disclosed
EP-0785926-A1 NEW CARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE BASF AKTIENGESELLSCHAFT (DE) 1997-07-30 EP disclosed
US-5559109-A Method of treating a PAF-mediated pathology or for treating or preventing psoriasis, nephritis, asthma or shock by administering a PAF antagonist SANKKO COMPANY, LIMITED (JP) 1996-09-24 US disclosed
US-5556852-A PLATELET ACTIVATING FACTOR ANTAGONISTS SANKYO COMPANY, LIMITED (JP) 1996-09-17 US disclosed
WO-1996011914-A1 NEW CARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE BASF AKTIENGESELLSCHAFT (DE) 1996-04-25 WO disclosed
US-5442071-A Photostability CIBA-GEIGY CORPORATION (US) 1995-08-15 US disclosed
US-5369106-A N-acryloylpiperazine derivatives, their preparation and their use of PAF antagonists SANKYO COMPANY, LIMITED (JP) 1994-11-29 US disclosed
US-5192766-A Platelet activating factor antagonist SANKYO COMPANY, LIMITED (JP) 1993-03-09 US disclosed
US-4595532-A N-(substituted-methyl)-azetidin-2-ones UNIVERSITY OF NOTRE DAME DU LAC (US) 1986-06-17 US disclosed
EP-0116432-A2 Improvements in or relating to N-(substituted-methyl)-azetidin-2-ones THE UNIVERSITY OF NOTRE DAME DU LAC (US) 1984-08-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210198235-A1 DERIVATIVES OF PIPERLONGUMINE AND USES THEREOF THPO, PIR, PAK6 MEN1 1394/4885KMT2A 2507/4885NPC1 868/4885
US-11485725-B2 Derivatives of piperlongumine and uses thereof PIR, THPO, DHPS MEN1 1372/4885KMT2A 2612/4885NPC1 768/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.