SCHEMBL10714432

SCHEMBL10714432

O=C(O)C(Sc1ccccc1)(C(=O)O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.45
FFAR1 O14842 1/20 0.39
CYP2D6 P10635 1/20 0.38
MAPT P10636 3/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 4/20 0.37
TSHR P16473 1/20 0.37
KCNN4 O15554 2/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HIF1A Q16665 1/20 0.36
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
HPGD P15428 3/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10880203 0.77 CYP1A2 (0.48) CYP1A2CYP2D6MAPTKMT2AALDH1A1
SCHEMBL3150010 0.71 SLC22A12 (0.50) FFAR1ALDH1A1HPGD
SCHEMBL21253178 0.71 CYP1A2 (0.46) CYP1A2FFAR1MAPTKMT2AALDH1A1
SCHEMBL15114537 0.71 CES1 (0.41) CYP1A2FFAR1MAPTALDH1A1TSHR
SCHEMBL28846242 0.69 MAPT (0.43) CYP1A2FFAR1MAPTALDH1A1TSHR
SCHEMBL11270832 0.69 KIF11 (0.43) MAPTALDH1A1TSHRKCNN4HPGD
SCHEMBL11208198 0.68 ALDH1A1 (0.47) FFAR1MAPTKMT2AALDH1A1TSHR
SCHEMBL7074813 0.68 CES1 (0.44) CYP1A2FFAR1MAPTALDH1A1TSHR
SCHEMBL11264686 0.68 ALDH1A1 (0.42) CYP1A2FFAR1CYP2D6MAPTKMT2A
SCHEMBL5552914 0.68 POLB (0.44) CYP1A2FFAR1MAPTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161932-B1 PREPARATION OF CARBOXYPHENYLTHIOPHENYLACETIC ACIDS MERCK & CO. INC. (US) 1988-04-13 EP claimed
EP-0161932-A2 Preparation of carboxyphenylthiophenylacetic acids MERCK & CO. INC. (US) 1985-11-21 EP claimed
EP-0161932-B1 PREPARATION OF CARBOXYPHENYLTHIOPHENYLACETIC ACIDS MERCK & CO. INC. (US) 1988-04-13 EP disclosed
EP-0161932-A2 Preparation of carboxyphenylthiophenylacetic acids MERCK & CO. INC. (US) 1985-11-21 EP disclosed
EP-0161932-A2 Preparation of carboxyphenylthiophenylacetic acids MERCK & CO. INC. (US) 1985-11-21 EP disclosed
EP-0161932-A2 Preparation of carboxyphenylthiophenylacetic acids MERCK & CO. INC. (US) 1985-11-21 EP disclosed