Citric Acid

Citric Acid

SCHEMBL10728752

C[N+](C)(C)CC(=O)O.C[N+](C)(C)CC(=O)O.O.O=C(O)CC(O)(CC(=O)O)C(=O)[O-].O=C(O)CC(O)(CC(=O)O)C(=O)[O-]

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACVR1ADORA1ADORA2AADORA2BADORA3ESR1ESR2FLT3GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSC1GSK3AGSK3BHRH1HRH2HTR7IDH1IDH2IMPA1IRAK1JAK1JAK2JAK3MEN1OPRM1P2RX3PDE5ASCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASIGMAR1SLC6A2SYKTACR1TOP2ATYK2

The experimentally established mechanism targets of Citric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.54
ALDH1A1 P00352 2/20 0.52
LMNA P02545 1/20 0.52
APEX1 P27695 1/20 0.52
CA4 P22748 1/20 0.43
HMGCR P04035 1/20 0.37
CHRM1 P11229 1/20 0.37
TBXA2R P21731 1/20 0.37
ADRA1A P35348 1/20 0.37
BBOX1 O75936 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
HIF1A Q16665 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Citric Acid SCHEMBL379527 0.98 TSHR (0.56) TSHRALDH1A1LMNAAPEX1CA4
Citric Acid SCHEMBL18584347 0.96 TSHR (0.54) TSHRALDH1A1LMNAAPEX1CA4
Citric Acid SCHEMBL7083476 0.88 CA4 (0.50) TSHRALDH1A1LMNAAPEX1CA4
Citric Acid SCHEMBL36782 0.86 CA4 (0.52) TSHRALDH1A1LMNAAPEX1CA4
Citric Acid SCHEMBL22229905 0.82 ALDH1A1 (0.65) TSHRALDH1A1LMNAAPEX1HMGCR
Citric Acid SCHEMBL3683509 0.81 ALDH1A1 (0.54) TSHRALDH1A1LMNAAPEX1CA4
Citric Acid SCHEMBL23320255 0.81 CA4 (0.56) TSHRALDH1A1CA4HMGCRCHRM1
Citric Acid SCHEMBL1092138 0.81 CA4 (0.64) TSHRALDH1A1CA4HMGCRCHRM1
Citric Acid SCHEMBL28287041 0.81 CA4 (0.64) TSHRALDH1A1CA4HMGCRCHRM1
Citric Acid SCHEMBL28164924 0.81 CA4 (0.64) TSHRALDH1A1CA4HMGCRCHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4703045-A BETAINE SALTS SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (FR) 1987-10-27 US disclosed
US-4593020-A Betaine citrate SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (FR) 1986-06-03 US disclosed