SCHEMBL10734451

SCHEMBL10734451

COc1ccc(C=C(NC(C)=O)C(=O)O)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
THRB P10828 1/20 0.51
ATM Q13315 1/20 0.51
GSK3B P49841 2/20 0.50
HDAC3 O15379 2/20 0.49
HDAC1 Q13547 2/20 0.49
HDAC2 Q92769 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
F3 P13726 2/20 0.49
BACE1 P56817 1/20 0.46
CYP1A2 P05177 1/20 0.46
KDM4E B2RXH2 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
AKR1C3 P42330 1/20 0.46
TRPM8 Q7Z2W7 1/20 0.46
HDAC4 P56524 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC10 Q969S8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28422488 1.00 ALDH1A1 (0.52) ALDH1A1THRBATMGSK3BHDAC3
SCHEMBL10734447 1.00 ALDH1A1 (0.52) ALDH1A1THRBATMGSK3BHDAC3
SCHEMBL8655219 0.87 ALDH1A1 (0.52) ALDH1A1THRBATMGSK3BHDAC3
SCHEMBL13906641 0.87 ALDH1A1 (0.52) ALDH1A1THRBATMGSK3BHDAC3
SCHEMBL11183020 0.86 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTCYP3A4SMN1; SMN2
SCHEMBL11719071 0.86 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTCYP3A4SMN1; SMN2
SCHEMBL14997267 0.82 THRB (0.49) ALDH1A1THRBATMGSK3BHDAC3
SCHEMBL8653627 0.82 ALDH1A1 (0.58) ALDH1A1CYP1A2KDM4EMAPTBCHE
SCHEMBL8653628 0.82 ALDH1A1 (0.58) ALDH1A1CYP1A2KDM4EMAPTBCHE
SCHEMBL10739476 0.81 ALDH1A1 (0.52) ALDH1A1GSK3BF3BACE1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4634775-A HYDROGENATION CATALYSTS FOR ACYLAMINO-ACRYLIC ACIDS DEGUSSA AKTIENGESELLSCHAFT (DE) 1987-01-06 US disclosed
EP-0151282-A1 Optically active 3,4-bis-(diphenylphosphino)-pyrrolidine, rhodium complexes containing them as chiral ligands, and their use Degussa Aktiengesellschaft (DE) 1985-08-14 EP disclosed