SCHEMBL10743370

SCHEMBL10743370

CC(=O)N(C)CN1CCN(c2ncccn2)CC1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.52
MDM2 Q00987 2/20 0.52
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
HRH3 Q9Y5N1 2/20 0.48
ALDH1A1 P00352 7/20 0.48
TDP1 Q9NUW8 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
HTR1A P08908 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48
TSHR P16473 1/20 0.47
HTT P42858 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
DRD2 P14416 2/20 0.45
DRD4 P21917 1/20 0.44
DRD3 P35462 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5538980 0.78 KDM4E (0.61) KDM4EMDM2NPC1RAB9AHRH3
SCHEMBL19658668 0.77 KDM4E (0.51) KDM4EMDM2NPC1RAB9AALDH1A1
SCHEMBL4500807 0.73 KDM4E (0.56) KDM4EMDM2NPC1RAB9AHRH3
SCHEMBL7356339 0.72 ALDH1A1 (0.66) KDM4EMDM2ALDH1A1TDP1SMN1; SMN2
SCHEMBL1919434 0.72 MEN1 (0.73) KDM4ENPC1RAB9AALDH1A1TSHR
SCHEMBL10332949 0.72 HRH3 (0.62) HRH3HTR1ADRD2DRD4DRD3
SCHEMBL10527898 0.72 HRH3 (0.52) KDM4EHRH3ALDH1A1TDP1SMN1; SMN2
SCHEMBL4406529 0.71 ALDH1A1 (0.60) KDM4EMDM2ALDH1A1TDP1SMN1; SMN2
Hydrochloric Acid SCHEMBL1371732 0.71 ALDH1A1 (0.64) KDM4EMDM2ALDH1A1TDP1SMN1; SMN2
SCHEMBL2633644 0.71 MEN1 (0.54) KDM4EMDM2ALDH1A1TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4668687-A Psychogeriatric 1-(2-pyrimidinyl)piperazinyl derivatives of 1-pyrrolidin-2-ones BRISTOL-MYERS COMPANY (US) 1987-05-26 US claimed