SCHEMBL10744375

SCHEMBL10744375

COc1cc(OS(C)(=O)=O)cc(-c2nc3ncccc3[nH]2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 6/20 0.65
PDE2A O00408 1/20 0.53
FGFR1 P11362 1/20 0.51
FGFR2 P21802 1/20 0.51
FGFR3 P22607 1/20 0.51
PDE5A O76074 3/20 0.48
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
HPGD P15428 1/20 0.46
KMT2A Q03164 1/20 0.46
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
HSD17B10 Q99714 1/20 0.46
PRMT5 O14744 2/20 0.45
HPSE Q9Y251 1/20 0.44
CYP2C9 P11712 1/20 0.43
NOS1 P29475 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10744129 0.81 AURKA (0.70) AURKAPDE2AFGFR1FGFR2FGFR3
SCHEMBL10748267 0.81 AURKA (0.57) AURKAPDE2APDE5AKDM4EMEN1
SCHEMBL10609325 0.80 PDE2A (0.77) AURKAPDE2APDE5AKDM4EMEN1
SCHEMBL9634492 0.78 AURKA (0.63) AURKAPDE2AFGFR1FGFR2FGFR3
SCHEMBL11772846 0.77 AURKA (1.00) AURKAPDE2APDE5AKDM4EALDH1A1
SCHEMBL709311 0.76 AURKA (0.54) AURKAPDE2APRMT5
SCHEMBL10984029 0.75 AURKA (0.80) AURKAPDE2AFGFR1FGFR2FGFR3
SCHEMBL10266345 0.75 AURKA (0.58) AURKAPDE2AFGFR1FGFR2FGFR3
SCHEMBL10746998 0.74 PDE2A (0.53) AURKAPDE2APDE5AKDM4EMEN1
SCHEMBL11775080 0.74 PDE2A (0.72) AURKAPDE2AFGFR1FGFR2FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4696931-A CARDIOVASCULAR DISORDERS, CARDIOTONIC AGENTS DR. KARL THOMAE GMBH (DE) 1987-09-29 US disclosed
US-4582837-A Imidazo[4,5-b] and [4,5-c]pyridine derivatives having cardiotonic activity DR. KARL THOMAE GMBH (DE) 1986-04-15 US disclosed
EP-0098448-A2 Imidazole derivatives, their preparation and medicines containing these compounds Dr. Karl Thomae GmbH (DE) 1984-01-18 EP disclosed