SCHEMBL10745014

SCHEMBL10745014

COCC(=O)c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSR P00390 2/20 0.56
MMP2 P08253 1/20 0.47
MMP9 P14780 1/20 0.47
MMP8 P22894 1/20 0.47
ENPP2 Q13822 1/20 0.45
AKR1C3 P42330 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1303853 0.82 ALDH1A1 (0.57) GSRMMP2MMP9MMP8ENPP2
SCHEMBL10541229 0.80 GSR (0.54) GSRMMP2MMP9MMP8ENPP2
SCHEMBL1303634 0.80 GSR (0.54) GSRMMP2MMP9MMP8
SCHEMBL5058142 0.79 GSR (0.61) GSRMMP2MMP9MMP8ENPP2
SCHEMBL1185872 0.79 GSR (0.61) GSRMMP2MMP9MMP8ENPP2
SCHEMBL15556865 0.77 GSR (0.59) GSRMMP2MMP9MMP8ENPP2
SCHEMBL28990483 0.77 GSR (0.59) GSRMMP2MMP9MMP8ENPP2
SCHEMBL125350 0.77 GSR (0.59) GSRMMP2MMP9MMP8ENPP2
SCHEMBL22584909 0.77 GSR (0.59) GSRMMP2MMP9MMP8ENPP2
SCHEMBL16923800 0.77 GSR (0.59) GSRMMP2MMP9MMP8ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4670445-A VASODILATORS ELI LILLY AND COMPANY (US) 1987-06-02 US disclosed
EP-0113236-B1 SUBSTITUTED IMIDAZOPYRIMIDINES-PYRAZINES, AND -TRIAZINES ELI LILLY AND COMPANY (US) 1987-04-22 EP disclosed
US-4636502-A Methods of producing a positive inotropic effect or vasodilation by administration of 2-phenyl imidazo pyrimidines and pyrazines ELI LILLY AND COMPANY (US) 1987-01-13 US disclosed
US-4578387-A VASODILATION; DERIVATIVES OF 2-PHENYL-5,6,7,8-TETRAHYDROIMADAZO/1,2-A/PYRAZINE ELI LILLY AND COMPANY (US) 1986-03-25 US disclosed
EP-0154494-A2 Phenylimidazole inotropic agents ELI LILLY AND COMPANY (US) 1985-09-11 EP disclosed
US-4537889-A PHENYL SUBSTITUTED IMIDAZO COMPOUNDS ELI LILLY AND COMPANY (US) 1985-08-27 US disclosed
EP-0113236-A1 Substituted imidazopyrimidines-pyrazines, and -triazines ELI LILLY AND COMPANY (US) 1984-07-11 EP disclosed