SCHEMBL5058142

SCHEMBL5058142

CS(=O)(=O)c1ccc(C(=O)CO)cc1

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSR P00390 2/20 0.61
MMP2 P08253 1/20 0.50
MMP9 P14780 1/20 0.50
MMP8 P22894 1/20 0.50
ENPP2 Q13822 1/20 0.50
AKR1C3 P42330 1/20 0.47
PTGS2 P35354 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1185872 0.83 GSR (0.61) GSRMMP2MMP9MMP8ENPP2
SCHEMBL10831304 0.82 GSR (0.59) GSRMMP2MMP9MMP8ENPP2
SCHEMBL8233398 0.82 GSR (0.59) GSRMMP2MMP9MMP8ENPP2
SCHEMBL22584909 0.82 GSR (0.59) GSRMMP2MMP9MMP8ENPP2
SCHEMBL16923800 0.82 GSR (0.59) GSRMMP2MMP9MMP8ENPP2
SCHEMBL125350 0.82 GSR (0.59) GSRMMP2MMP9MMP8ENPP2
SCHEMBL15556865 0.82 GSR (0.59) GSRMMP2MMP9MMP8ENPP2
SCHEMBL28990483 0.82 GSR (0.59) GSRMMP2MMP9MMP8ENPP2
Hydrochloric Acid SCHEMBL15465891 0.80 GSR (0.60) GSRMMP2MMP9MMP8ENPP2
SCHEMBL25876517 0.80 GSR (0.57) GSRMMP2MMP9MMP8ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4387617-A1 ACID CERAMIDASE INHIBITORS AND USES THEREOF The Regents of the University of California (US) 2024-06-26 EP disclosed
WO-2023023156-A1 ACID CERAMIDASE INHIBITORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-02-23 WO disclosed
WO-2023023156-A1 ACID CERAMIDASE INHIBITORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-02-23 WO disclosed
CN-110015983-A 1,2- dicarbapentaborane class compound and its synthetic method 华东师范大学 2019-07-16 CN disclosed
US-20080044350-A1 Optical Imaging Contrast Agents for Imaging Lung Cancer GE HEALTHCARE AS (NO) 2008-02-21 US disclosed
US-20080044350-A1 Optical Imaging Contrast Agents for Imaging Lung Cancer GE HEALTHCARE AS (NO) 2008-02-21 US disclosed
US-20080044350-A1 Optical Imaging Contrast Agents for Imaging Lung Cancer GE HEALTHCARE AS (NO) 2008-02-21 US disclosed
US-20070212305-A1 Optical Imaging Contrast Agents For Imaging Lung Cancer AMERSHAM HEALTH AS (NO) 2007-09-13 US disclosed
US-20070212305-A1 Optical Imaging Contrast Agents For Imaging Lung Cancer AMERSHAM HEALTH AS (NO) 2007-09-13 US disclosed
US-20070212305-A1 Optical Imaging Contrast Agents For Imaging Lung Cancer AMERSHAM HEALTH AS (NO) 2007-09-13 US disclosed
EP-1667734-A2 OPTICAL IMAGING OF COLORECTAL CANCER GE Healthcare AS (NO) 2006-06-14 EP disclosed
WO-2005058370-A1 OPTICAL IMAGING CONTRAST AGENTS FOR IMAGING LUNG CANCER AMERSHAM HEALTH AS (NO) 2005-06-30 WO disclosed
WO-2005058372-A1 OPTICAL IMAGING CONTRAST AGENTS FOR IMAGING LUNG CANCER AMERSHAM HEALTH AS (NO) 2005-06-30 WO disclosed
WO-2005030266-A2 OPTICAL IMAGING OF COLORECTAL CANCER AMERSHAM HEALTH AS (NO) 2005-04-07 WO disclosed
US-6869968-B1 Such as 3-(4-fluorophenyl)-4-(4-methysulphonylphenyl)-2-(3H)-oxazolone; for treating colorectal cancer, fevers, and inflammation ALLMIRALL PRODESFARMA S.A. (ES) 2005-03-22 US disclosed
EP-0888316-B1 2-(3H)-OXAZOLONE DERIVATIVES AND THEIR USE AS COX-2 INHIBITORS ALMIRALL PRODESFARMA SA (ES) 2000-11-02 EP disclosed
EP-1017685-A1 NEW 2-(3H)-OXAZOLONE DERIVATIVES ALMIRALL-PRODESFARMA, S.A. (ES) 2000-07-12 EP disclosed
WO-1999014205-A1 NEW 2-(3H)-OXAZOLONE DERIVATIVES ALMIRALL PRODESFARMA S.A. (ES) 1999-03-25 WO disclosed
EP-0888316-A1 2-(3H)-OXAZOLONE DERIVATIVES AND THEIR USE AS COX-2 INHIBITORS ALMIRALL-PRODESFARMA, S.A. (ES) 1999-01-07 EP disclosed
WO-1997034882-A1 2-(3H)-OXAZOLONE DERIVATIVES AND THEIR USE AS COX-2 INHIBITORS ALMIRALL PRODESFARMA, S.A. (ES) 1997-09-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080044350-A1 Optical Imaging Contrast Agents for Imaging Lung Cancer KLK3, ROCK1, SMO GSR 1819/4885MMP2 2528/4885MMP9 709/4885
US-20070212305-A1 Optical Imaging Contrast Agents For Imaging Lung Cancer IQGAP1, AQP3, ROCK1 GSR 2863/4885MMP2 2845/4885MMP9 909/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.