SCHEMBL10745643

SCHEMBL10745643

c1ccc(CCOc2ccccc2-c2cn3c(n2)CCCC3)cc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 8/20 0.51
ALDH1A1 P00352 3/20 0.48
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
LMNA P02545 3/20 0.45
HTT P42858 2/20 0.45
KDM4E B2RXH2 1/20 0.45
HRH3 Q9Y5N1 1/20 0.44
TP53 P04637 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
IDO1 P14902 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
TNF P01375 1/20 0.38
ABCB1 P08183 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10745646 0.81 WDR5 (0.73) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL10747411 0.81 WDR5 (0.42) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL10750669 0.79 WDR5 (0.53) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL10745635 0.74 WDR5 (0.48) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL219606 0.72 WDR5 (0.56) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL21484047 0.71 WDR5 (0.52) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL4839937 0.71 WDR5 (0.90) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL10750608 0.70 ALDH1A1 (0.51) WDR5ALDH1A1NPC1RAB9ALMNA
SCHEMBL2813551 0.70 PDCD1 (0.57) WDR5IDO1
SCHEMBL10747533 0.68 HRH3 (0.40) WDR5ALDH1A1NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4670445-A VASODILATORS ELI LILLY AND COMPANY (US) 1987-06-02 US disclosed
US-4578387-A VASODILATION; DERIVATIVES OF 2-PHENYL-5,6,7,8-TETRAHYDROIMADAZO/1,2-A/PYRAZINE ELI LILLY AND COMPANY (US) 1986-03-25 US disclosed