SCHEMBL1074656

SCHEMBL1074656

O=S(=O)(Cl)c1cccc(-c2nccs2)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KAT6A Q92794 1/20 0.52
PDPK1 O15530 1/20 0.51
CYP2A6 P11509 1/20 0.46
LOXL2 Q9Y4K0 1/20 0.42
ACLY P53396 2/20 0.42
ALDH1A1 P00352 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
FFAR1 O14842 1/20 0.40
GPR119 Q8TDV5 1/20 0.39
HDAC2 Q92769 1/20 0.38
PIP4K2C Q8TBX8 2/20 0.37
VCP P55072 1/20 0.37
NTRK1 P04629 1/20 0.36
ADRB2 P07550 1/20 0.36
PRKDC P78527 1/20 0.36
SYK P43405 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1668053 0.84 KAT6A (0.52) KAT6APDPK1CYP2A6LOXL2
SCHEMBL12658214 0.84 KAT6A (0.52) KAT6APDPK1CYP2A6LOXL2PIP4K2C
Hydrochloric Acid SCHEMBL5692827 0.83 KAT6A (0.51) KAT6APDPK1CYP2A6LOXL2
Hydrochloric Acid SCHEMBL5692840 0.83 KAT6A (0.51) KAT6APDPK1CYP2A6LOXL2
SCHEMBL15805858 0.79 PDPK1 (0.72) KAT6APDPK1CYP2A6LOXL2PTGDR2
SCHEMBL21999853 0.78 ACLY (0.50) KAT6APDPK1CYP2A6LOXL2ACLY
SCHEMBL16159287 0.76 PDPK1 (0.67) KAT6APDPK1CYP2A6LOXL2PTGDR2
SCHEMBL10408548 0.75 ALDH1A1 (0.56) ALDH1A1HSD17B10TDP1
SCHEMBL996104 0.75 ALDH1A1 (0.48) KAT6ACYP2A6ALDH1A1HSD17B10TDP1
SCHEMBL468088 0.75 PDPK1 (0.60) KAT6APDPK1CYP2A6LOXL2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274296-A1 HYDROXYMETHYL PYRROLIDINES AS BETA 3 ADRENERGIC RECEPTOR AGONISTS Merck Sharp & Dohme Corp. (US) 2011-01-19 EP disclosed